SCHEMBL28705205

SCHEMBL28705205

O=C(O)c1nc(-c2ccccc2)cn1Cc1ccccc1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 4/20 0.49
GAA P10253 1/20 0.44
PKM P14618 1/20 0.44
TSHR P16473 1/20 0.44
CYP19A1 P11511 1/20 0.44
ADORA2A P29274 1/20 0.43
TLR8 Q9NR97 2/20 0.42
NOTUM Q6P988 1/20 0.42
MEN1 O00255 2/20 0.42
KMT2A Q03164 2/20 0.42
CASP3 P42574 1/20 0.42
SENP8 Q96LD8 1/20 0.42
SENP7 Q9BQF6 1/20 0.42
SENP6 Q9GZR1 1/20 0.42
LMNA P02545 1/20 0.41
DHODH Q02127 1/20 0.41
CCNC P24863 1/20 0.41
CDK8 P49336 1/20 0.41
IDO1 P14902 1/20 0.41
CYP11B1 P15538 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6861398 0.83 TLR8 (0.50) PKMCYP19A1ADORA2ATLR8DHODH
SCHEMBL28710551 0.79 NOTUM (0.50) BRD4GAAPKMTSHRCYP19A1
SCHEMBL28706154 0.78 NPSR1 (0.42) BRD4GAAPKMTSHRCYP19A1
SCHEMBL28027825 0.77 BRD4 (0.64) BRD4GAACYP19A1ADORA2ATLR8
SCHEMBL2337948 0.77 BRD4 (0.48) BRD4CYP19A1ADORA2ATLR8NOTUM
SCHEMBL15135930 0.76 TUBB4A (0.48)
SCHEMBL2337941 0.76 PDE10A (0.47) BRD4TSHRCYP19A1ADORA2ALMNA
SCHEMBL28426192 0.76 TLR8 (0.60) BRD4PKMCYP19A1ADORA2ATLR8
SCHEMBL28717264 0.76 BRD4 (0.49) BRD4GAACYP19A1ADORA2ATLR8
SCHEMBL1927995 0.73 PDE10A (0.47) BRD4GAAPKMCYP19A1ADORA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114230522-A Imidazole-2-carboxylic acid metal beta-lactamase inhibitor and preparation method and application thereof 四川大学 2022-03-25 CN disclosed