SCHEMBL28708176

SCHEMBL28708176

O=C(C=Cc1cccs1)c1ccc(O)cc1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ABCG2 Q9UNQ0 2/20 1.00
MAPT P10636 9/20 0.74
NPC1 O15118 2/20 0.62
RAB9A P51151 2/20 0.62
CASP3 P42574 1/20 0.62
SENP8 Q96LD8 1/20 0.62
SENP7 Q9BQF6 1/20 0.62
SENP6 Q9GZR1 1/20 0.62
MEN1 O00255 5/20 0.59
KMT2A Q03164 5/20 0.59
LMNA P02545 4/20 0.59
CYP3A4 P08684 3/20 0.59
CYP2C9 P11712 1/20 0.59
CYP2C19 P33261 1/20 0.59
HCAR2 Q8TDS4 1/20 0.59
F3 P13726 2/20 0.56
MAOA P21397 2/20 0.56
MAOB P27338 2/20 0.56
TDP1 Q9NUW8 2/20 0.56
ALDH2 P05091 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17429547 1.00 ABCG2 (1.00) ABCG2MAPTNPC1RAB9ACASP3
SCHEMBL11477087 0.87 ABCG2 (0.77) ABCG2MAPTNPC1RAB9ACASP3
SCHEMBL11477089 0.87 ABCG2 (0.77) ABCG2MAPTNPC1RAB9ACASP3
SCHEMBL8078718 0.86 ABCG2 (0.76) ABCG2MAPTNPC1RAB9ACASP3
SCHEMBL8663226 0.86 ABCG2 (0.76) ABCG2MAPTNPC1RAB9ACASP3
SCHEMBL3035768 0.85 ABCG2 (0.74) ABCG2MAPTNPC1RAB9ACASP3
SCHEMBL7203615 0.85 MAPT (1.00) ABCG2MAPTNPC1RAB9ACASP3
SCHEMBL7203616 0.85 MAPT (1.00) ABCG2MAPTNPC1RAB9ACASP3
SCHEMBL3035766 0.85 ABCG2 (0.74) ABCG2MAPTNPC1RAB9ACASP3
SCHEMBL31301136 0.85 ABCG2 (0.74) ABCG2MAPTNPC1RAB9ACASP3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116217461-B Chalcone derivative containing indole structure and preparation method and application thereof 贵州大学 2024-10-18 CN disclosed
CN-116283789-B Pyridazine-containing chalcone derivative and preparation method and application thereof 贵州大学 2024-09-03 CN disclosed
CN-116283789-A Pyridazine-containing chalcone derivative and preparation method and application thereof 贵州大学 2023-06-23 CN disclosed
CN-116217461-A Chalcone derivative containing indole structure and preparation method and application thereof 贵州大学 2023-06-06 CN disclosed
CN-114085199-B Chalcone derivative containing sulfonyl piperazine as well as preparation method and application thereof 贵州大学 2023-04-21 CN disclosed
CN-109293616-B Coumarin-containing chalcone derivatives, and preparation method and application thereof 贵州大学 2022-06-21 CN disclosed
CN-109810068-B Chalcone derivative containing thioether triazole, preparation method and application 贵州大学 2022-03-18 CN disclosed
CN-114085199-A Chalcone derivative containing sulfonyl piperazine and preparation method and application thereof 贵州大学 2022-02-25 CN disclosed