SCHEMBL2870826

SCHEMBL2870826

CC1(C)OB(c2cccc3cc(-c4ccnc(NCCN5CCNC5=O)n4)sc23)OC1(C)C

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BRAF P15056 7/20 0.40
IRAK1 P51617 1/20 0.39
IRAK4 Q9NWZ3 1/20 0.39
RAF1 P04049 6/20 0.38
MAPK3 P27361 1/20 0.35
MAPK1 P28482 1/20 0.35
MKNK1 Q9BUB5 2/20 0.34
EGFR P00533 1/20 0.34
IKBKB O14920 1/20 0.33
CHUK O15111 1/20 0.33
IKBKG Q9Y6K9 1/20 0.33
ADORA2A P29274 1/20 0.33
ADORA1 P30542 1/20 0.33
EIF2AK2 P19525 3/20 0.33
SCN9A Q15858 2/20 0.33
CDK4 P11802 1/20 0.32
CCND1 P24385 1/20 0.32
ERN1 O75460 1/20 0.32
ABL1 P00519 1/20 0.32
FGFR1 P11362 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL388682 0.87 IRAK1 (0.39) BRAFIRAK1IRAK4RAF1ADORA2A
SCHEMBL2873640 0.87 IRAK1 (0.39) BRAFIRAK1IRAK4RAF1MAPK3
SCHEMBL2870590 0.86 IRAK1 (0.39) BRAFIRAK1IRAK4RAF1MAPK3
SCHEMBL2879156 0.82 BRAF (0.45) BRAFIRAK1IRAK4RAF1MKNK1
SCHEMBL2972101 0.78 IKBKB (0.50) BRAFIRAK1IRAK4RAF1IKBKB
SCHEMBL389292 0.77 BRAF (0.46) BRAFIRAK1IRAK4RAF1MAPK1
SCHEMBL393624 0.77 BRAF (0.42) BRAFIRAK1IRAK4RAF1MKNK1
SCHEMBL391684 0.77 BRAF (0.41) BRAFIRAK1IRAK4RAF1MKNK1
SCHEMBL1336964 0.77 BRAF (0.41) BRAFIRAK1IRAK4RAF1MKNK1
SCHEMBL391913 0.76 BRAF (0.42) BRAFIRAK1IRAK4RAF1MKNK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2125794-B1 IMIDAZOLIDINONYL AMINOPYRIMIDINE COMPOUNDS FOR THE TREATMENT OF CANCER LILLY CO ELI (US) 2010-10-20 EP disclosed