SCHEMBL2879156

SCHEMBL2879156

O=C1NCCN1CCNc1nccc(-c2cc3cccc(Br)c3s2)n1

nearest known ligand 0.45

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
BRAF P15056 8/20 0.45
RAF1 P04049 7/20 0.41
IRAK1 P51617 1/20 0.38
IRAK4 Q9NWZ3 1/20 0.38
IKBKB O14920 2/20 0.37
CHUK O15111 2/20 0.37
IKBKG Q9Y6K9 2/20 0.37
SCN9A Q15858 5/20 0.36
ADORA2A P29274 1/20 0.35
ADORA1 P30542 1/20 0.35
MKNK1 Q9BUB5 2/20 0.35
EIF2AK2 P19525 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL388891 0.85 SCN9A (0.42) BRAFRAF1IRAK1IRAK4SCN9A
SCHEMBL2972101 0.85 IKBKB (0.50) BRAFRAF1IRAK1IRAK4IKBKB
SCHEMBL391325 0.84 BRAF (0.41) BRAFRAF1IRAK1IRAK4SCN9A
SCHEMBL2923633 0.84 IRAK1 (0.40) BRAFRAF1IRAK1IRAK4SCN9A
SCHEMBL389292 0.84 BRAF (0.46) BRAFRAF1IRAK1IRAK4IKBKB
SCHEMBL2878585 0.83 IRAK1 (0.39) BRAFRAF1IRAK1IRAK4SCN9A
SCHEMBL392544 0.82 BRAF (0.42) BRAFRAF1IRAK1IRAK4IKBKB
SCHEMBL391913 0.82 BRAF (0.42) BRAFRAF1IRAK1IRAK4IKBKB
SCHEMBL2870826 0.82 BRAF (0.40) BRAFRAF1IRAK1IRAK4IKBKB
SCHEMBL2984342 0.82 BRAF (0.50) BRAFRAF1IRAK1IRAK4SCN9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2125794-B1 IMIDAZOLIDINONYL AMINOPYRIMIDINE COMPOUNDS FOR THE TREATMENT OF CANCER LILLY CO ELI (US) 2010-10-20 EP disclosed
EP-2125793-B1 IMIDAZOLIDINONYL AMINOPYRIMIDINE COMPOUNDS FOR THE TREATMENT OF CANCER LILLY CO ELI (US) 2010-09-01 EP disclosed