SCHEMBL28709090

SCHEMBL28709090

c1ccc2nc(OCCCCN3CCN(c4cccc5sccc45)CC3)ccc2c1

nearest known ligand 0.69

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 6/20 0.64
DRD2 P14416 6/20 0.64
HTR2A P28223 6/20 0.64
HTR2C P28335 2/20 0.58
ADRA1A P35348 2/20 0.58
HRH1 P35367 2/20 0.58
ADRB2 P07550 1/20 0.58
ADRB1 P08588 1/20 0.58
ADRA2A P08913 1/20 0.58
ADRA2B P18089 1/20 0.58
ADRA2C P18825 1/20 0.58
DRD1 P21728 1/20 0.58
DRD4 P21917 1/20 0.58
DRD5 P21918 1/20 0.58
SLC6A2 P23975 1/20 0.58
ADRA1D P25100 1/20 0.58
HTR1D P28221 1/20 0.58
HTR1B P28222 1/20 0.58
HTR1E P28566 1/20 0.58
SLC6A4 P31645 1/20 0.58

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19549054 0.90 HTR1A (0.68) HTR1ADRD2HTR2AHTR2CADRA1A
SCHEMBL29433200 0.90 HTR1A (0.68) HTR1ADRD2HTR2AHTR2CADRA1A
SCHEMBL29242379 0.89 HTR1A (0.62) HTR1ADRD2HTR2AHTR2CADRA1A
SCHEMBL30901141 0.86 HTR1A (0.59) HTR1ADRD2HTR2AHTR2CADRA1A
SCHEMBL29242356 0.86 HTR1A (0.59) HTR1ADRD2HTR2AHTR2CADRA1A
SCHEMBL17765537 0.85 HTR1A (0.54) HTR1ADRD2HTR2AHTR2CADRA1A
SCHEMBL20021850 0.84 HTR1A (0.61) HTR1ADRD2HTR2AHTR2CADRA1A
SCHEMBL16443220 0.83 HTR1A (0.65) HTR1ADRD2HTR2AHTR2CADRA1A
SCHEMBL16443221 0.83 HTR1A (0.65) HTR1ADRD2HTR2AHTR2CADRA1A
SCHEMBL16442962 0.83 HTR1A (0.62) HTR1ADRD2HTR2AHTR2CADRA1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114166960-B Method for detecting substances related to epipiprazole 西安远大科创医药科技有限公司 2023-09-29 CN claimed
CN-114166960-A Detection method of brexpiprazole related substance 西安远大科创医药科技有限公司 2022-03-11 CN claimed
CN-114166960-B Method for detecting substances related to epipiprazole 西安远大科创医药科技有限公司 2023-09-29 CN disclosed
CN-114166960-A Detection method of brexpiprazole related substance 西安远大科创医药科技有限公司 2022-03-11 CN disclosed