SCHEMBL28709093

SCHEMBL28709093

CC(C)(C)OC(=O)N1CC=C(c2ccnc(N)c2)C1

nearest known ligand 0.43

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
TBK1 Q9UHD2 2/20 0.43
UCHL1 P09936 1/20 0.42
NR1H2 P55055 1/20 0.41
PDK4 Q16654 1/20 0.41
GRM1 Q13255 5/20 0.41
GRM5 P41594 5/20 0.41
WNT3A P56704 1/20 0.41
NAMPT P43490 1/20 0.41
TNK2 Q07912 2/20 0.41
BTK Q06187 1/20 0.40
CDK9 P50750 2/20 0.40
CYP11B2 P19099 1/20 0.39
CCNT1 O60563 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28471545 0.86 GRM1 (0.46) TBK1PDK4GRM1GRM5WNT3A
SCHEMBL26074128 0.86 GRM5 (0.43) TBK1PDK4GRM1GRM5WNT3A
SCHEMBL30545737 0.86 GRM5 (0.43) TBK1PDK4GRM1GRM5WNT3A
SCHEMBL31705477 0.84 WNT3A (0.42) TBK1NR1H2PDK4GRM1GRM5
SCHEMBL31704807 0.84 WNT3A (0.42) TBK1NR1H2PDK4GRM1GRM5
SCHEMBL24791833 0.84 WNT3A (0.42) TBK1PDK4GRM1GRM5WNT3A
SCHEMBL609042 0.83 NAMPT (0.44) NR1H2PDK4GRM1GRM5NAMPT
SCHEMBL29538449 0.83 NAMPT (0.44) NR1H2PDK4GRM1GRM5NAMPT
SCHEMBL19992989 0.82 GRM1 (0.56) PDK4GRM1GRM5NAMPT
SCHEMBL17002448 0.80 NR1H2 (0.52) NR1H2PDK4GRM1GRM5NAMPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114181257-A Pyridine compound, pharmaceutical composition containing pyridine compound, preparation method and application of pyridine compound 四川科伦博泰生物医药股份有限公司 2022-03-15 CN disclosed