SCHEMBL28709129

SCHEMBL28709129

COc1ccc(C(NC(=O)C(c2ccccc2)c2ccccc2)C(=O)NO)cc1

nearest known ligand 0.63

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CNR2 P34972 2/20 0.58
CNR1 P21554 1/20 0.58
HDAC3 O15379 1/20 0.56
HDAC4 P56524 1/20 0.56
HDAC1 Q13547 1/20 0.56
HDAC7 Q8WUI4 1/20 0.56
HDAC2 Q92769 1/20 0.56
HDAC10 Q969S8 1/20 0.56
HDAC11 Q96DB2 1/20 0.56
HDAC8 Q9BY41 1/20 0.56
HDAC6 Q9UBN7 1/20 0.56
HDAC9 Q9UKV0 1/20 0.56
HDAC5 Q9UQL6 1/20 0.56
ALDH1A1 P00352 2/20 0.54
NPSR1 Q6W5P4 1/20 0.54
KLK7 P49862 2/20 0.50
GPR88 Q9GZN0 1/20 0.50
ANPEP P15144 1/20 0.49
ATM Q13315 1/20 0.49
TP53 P04637 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28709128 1.00 CNR2 (0.58) CNR2CNR1HDAC3HDAC4HDAC1
SCHEMBL28785765 0.90 HDAC4 (0.70) CNR2CNR1HDAC3HDAC4HDAC1
SCHEMBL2841700 0.85 HDAC3 (0.64) CNR2CNR1HDAC3HDAC4HDAC1
SCHEMBL20490426 0.83 HDAC3 (0.60) CNR2CNR1HDAC3HDAC4HDAC1
SCHEMBL20490505 0.82 HDAC3 (0.58) CNR2CNR1HDAC3HDAC4HDAC1
SCHEMBL28709110 0.80 ANPEP (0.46) CNR2CNR1ALDH1A1NPSR1GPR88
SCHEMBL28710172 0.80 ANPEP (0.46) CNR2CNR1ALDH1A1NPSR1GPR88
SCHEMBL2843919 0.79 MAPK1 (0.56) CNR2CNR1HDAC3HDAC4HDAC1
SCHEMBL28934074 0.79 HDAC3 (0.51) CNR2CNR1HDAC3HDAC4HDAC1
SCHEMBL28934073 0.79 HDAC3 (0.51) CNR2CNR1HDAC3HDAC4HDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114181116-B D-amino acid derivative aminopeptidase N inhibitor, and preparation method and application thereof 山东中医药大学 2023-05-23 CN disclosed
CN-114181116-A D-amino acid derivative aminopeptidase N inhibitor and preparation method and application thereof 山东中医药大学 2022-03-15 CN disclosed