SCHEMBL28934073

SCHEMBL28934073

COc1ccc([C@@H](NC(=O)C(C)(c2ccccc2)c2ccccc2)C(=O)NO)cc1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC3 O15379 1/20 0.51
HDAC4 P56524 1/20 0.51
HDAC1 Q13547 1/20 0.51
HDAC7 Q8WUI4 1/20 0.51
HDAC2 Q92769 1/20 0.51
HDAC10 Q969S8 1/20 0.51
HDAC11 Q96DB2 1/20 0.51
HDAC8 Q9BY41 1/20 0.51
HDAC6 Q9UBN7 1/20 0.51
HDAC9 Q9UKV0 1/20 0.51
HDAC5 Q9UQL6 1/20 0.51
NPSR1 Q6W5P4 1/20 0.48
MMP1 P03956 4/20 0.47
ANPEP P15144 3/20 0.46
MMP3 P08254 2/20 0.45
MMP13 P45452 2/20 0.45
TNF P01375 1/20 0.45
MMP2 P08253 1/20 0.45
ADAM17 P78536 1/20 0.45
CNR2 P34972 3/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28934074 1.00 HDAC3 (0.51) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL28709110 0.88 ANPEP (0.46) NPSR1MMP1ANPEPMMP3MMP13
SCHEMBL28710172 0.88 ANPEP (0.46) NPSR1MMP1ANPEPMMP3MMP13
SCHEMBL28700696 0.80 CNR2 (0.48) HDAC1HDAC7MMP1ANPEPMMP3
SCHEMBL28700697 0.80 CNR2 (0.48) HDAC1HDAC7MMP1ANPEPMMP3
SCHEMBL28709128 0.79 CNR2 (0.58) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL28709129 0.79 CNR2 (0.58) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL28933993 0.77 ATM (0.54) NPSR1CNR2GPR88ATMTP53
SCHEMBL7036247 0.74 NPSR1 (0.69) NPSR1ANPEPCNR2ATMCNR1
SCHEMBL28785765 0.73 HDAC4 (0.70) HDAC3HDAC4HDAC1HDAC7HDAC2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114181116-B D-amino acid derivative aminopeptidase N inhibitor, and preparation method and application thereof 山东中医药大学 2023-05-23 CN disclosed
CN-114181116-A D-amino acid derivative aminopeptidase N inhibitor and preparation method and application thereof 山东中医药大学 2022-03-15 CN disclosed