SCHEMBL28711992

SCHEMBL28711992

c1cc(-c2csc(-c3csc(Nc4ccc5c(c4)OCO5)n3)n2)ccn1

nearest known ligand 0.73

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 6/20 0.73
ALOX5 P09917 2/20 0.70
CYP1A1 P04798 4/20 0.69
CYP1A2 P05177 4/20 0.69
CYP1B1 Q16678 4/20 0.69
MAPT P10636 5/20 0.68
SMN1; SMN2 Q16637 5/20 0.68
MEN1 O00255 3/20 0.68
ALDH1A1 P00352 3/20 0.68
KMT2A Q03164 3/20 0.68
TSHR P16473 2/20 0.68
NPC1 O15118 2/20 0.68
RAB9A P51151 2/20 0.68
HSD17B10 Q99714 1/20 0.68
LMNA P02545 2/20 0.61
GAA P10253 2/20 0.61
ROCK1 Q13464 1/20 0.54
CFTR P13569 1/20 0.54
MAPK1 P28482 1/20 0.53
POLB P06746 2/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1885662 0.94 PTGS2 (0.81) PTGS2ALOX5CYP1A1CYP1A2CYP1B1
SCHEMBL29654152 0.88 PTGS2 (0.69) PTGS2ALOX5CYP1A1CYP1A2CYP1B1
SCHEMBL28701603 0.88 PTGS2 (0.69) PTGS2ALOX5CYP1A1CYP1A2CYP1B1
SCHEMBL12298228 0.84 SMN1; SMN2 (0.93) PTGS2ALOX5CYP1A1CYP1A2CYP1B1
SCHEMBL28707160 0.84 CYP1A1 (0.68) PTGS2ALOX5CYP1A1CYP1A2CYP1B1
SCHEMBL207468 0.82 PTGS2 (0.77) PTGS2ALOX5CYP1A1CYP1A2CYP1B1
SCHEMBL28713936 0.81 CYP1A1 (1.00) PTGS2ALOX5CYP1A1CYP1A2CYP1B1
SCHEMBL12297517 0.81 SMN1; SMN2 (1.00) PTGS2ALOX5CYP1A1CYP1A2CYP1B1
SCHEMBL12298248 0.81 SMN1; SMN2 (1.00) PTGS2ALOX5CYP1A1CYP1A2CYP1B1
SCHEMBL12297293 0.80 PTGS2 (0.67) PTGS2ALOX5CYP1A1CYP1A2CYP1B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114249702-A N-aryl- [2,4 '-bithiazole ] -2' -amine compound and preparation and application thereof 沈阳药科大学 2022-03-29 CN disclosed