SCHEMBL28721995

SCHEMBL28721995

Brc1cccc2ccc(-c3cccnc3)nc12

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 5/20 0.51
BACE1 P56817 1/20 0.47
NPC1 O15118 2/20 0.47
HSP90AA1 P07900 1/20 0.46
HSP90AB1 P08238 1/20 0.46
PTK2 Q05397 1/20 0.46
ALDH1A1 P00352 2/20 0.45
CYP3A4 P08684 2/20 0.45
CYP1A2 P05177 1/20 0.45
CYP11B1 P15538 2/20 0.45
CYP11B2 P19099 2/20 0.45
CYP19A1 P11511 4/20 0.45
CYP17A1 P05093 1/20 0.45
MAPT P10636 2/20 0.44
KDM4E B2RXH2 1/20 0.44
LMNA P02545 1/20 0.44
TP53 P04637 1/20 0.44
HPGD P15428 1/20 0.44
ALOX15 P16050 1/20 0.44
HTT P42858 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29496195 1.00 CYP2A6 (0.51) CYP2A6BACE1NPC1HSP90AA1HSP90AB1
SCHEMBL28722905 0.83 RAB9A (0.53) BACE1NPC1CYP3A4CYP1A2CYP19A1
SCHEMBL29496146 0.83 BACE1 (0.50) CYP2A6BACE1NPC1HSP90AA1CYP3A4
SCHEMBL29496334 0.83 RAB9A (0.53) BACE1NPC1CYP3A4CYP1A2CYP19A1
SCHEMBL28722848 0.83 BACE1 (0.50) CYP2A6BACE1NPC1HSP90AA1CYP3A4
SCHEMBL15229057 0.82 PARP1 (0.54) BACE1NPC1ALDH1A1CYP3A4CYP1A2
SCHEMBL1030196 0.80 HSP90AA1 (0.54) CYP2A6NPC1HSP90AA1HSP90AB1PTK2
SCHEMBL19768555 0.79 CYP3A4 (0.57) CYP2A6NPC1HSP90AA1HSP90AB1PTK2
SCHEMBL14884092 0.79 NPC1 (0.59) CYP2A6NPC1HSP90AA1HSP90AB1PTK2
SCHEMBL28722873 0.79 BACE1 (0.46) BACE1NPC1HSP90AA1CYP3A4CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114269730-A 5-heteroaryl-pyridin-2-amine compounds as neuropeptide FF receptor antagonists 多曼治疗学公司 2022-04-01 CN disclosed