SCHEMBL28724766

SCHEMBL28724766

N#C/C=C(\C#N)c1cccc(Cl)c1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 6/20 0.52
ALDH1A1 P00352 3/20 0.52
NPC1 O15118 1/20 0.52
RAB9A P51151 1/20 0.52
NPSR1 Q6W5P4 1/20 0.52
HPGD P15428 2/20 0.46
LMNA P02545 2/20 0.46
CYP1A2 P05177 1/20 0.46
CYP2C9 P11712 1/20 0.46
CYP2C19 P33261 1/20 0.46
RECQL P46063 1/20 0.46
KMT2A Q03164 3/20 0.43
KDM4E B2RXH2 2/20 0.43
POLB P06746 2/20 0.43
PKM P14618 1/20 0.43
PARP1 P09874 1/20 0.43
HTT P42858 3/20 0.40
GABRA1 P14867 2/20 0.40
GABRG2 P18507 2/20 0.40
GABRB3 P28472 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29483451 1.00 MAPT (0.52) MAPTALDH1A1NPC1RAB9ANPSR1
SCHEMBL5865765 0.87 PDE4A (0.42) MAPTALDH1A1NPC1RAB9ANPSR1
SCHEMBL5865766 0.87 PDE4A (0.42) MAPTALDH1A1NPC1RAB9ANPSR1
SCHEMBL14156069 0.84 MAPT (0.54) MAPTALDH1A1NPC1RAB9ANPSR1
SCHEMBL7477836 0.80 PARP1 (0.44) MAPTALDH1A1NPC1RAB9ANPSR1
SCHEMBL8743683 0.80 CA12 (0.42) MAPTALDH1A1RAB9ANPSR1LMNA
SCHEMBL7477831 0.80 PARP1 (0.44) MAPTALDH1A1NPC1RAB9ANPSR1
SCHEMBL11123552 0.79 PARP1 (0.52) MAPTALDH1A1NPC1RAB9ANPSR1
SCHEMBL11072261 0.79 PARP1 (0.52) MAPTALDH1A1NPC1RAB9ANPSR1
SCHEMBL11072258 0.79 PARP1 (0.52) MAPTALDH1A1NPC1RAB9ANPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114349703-B Trifluoromethyl-4-cyano pyrazole compound, and preparation method and application thereof 天津大学 2024-05-10 CN disclosed
CN-114349703-A Trifluoromethyl-4-cyanopyrazole compound, and preparation method and application thereof 天津大学 2022-04-15 CN disclosed