SCHEMBL28740145

SCHEMBL28740145

Cc1nc(NC2CCCC2)c2ncn([C@@H]3O[C@H](C[O])[C@@H](O)[C@@H]3F)c2n1

nearest known ligand 0.59

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
NT5E P21589 6/20 0.59
ADORA3 P0DMS8 5/20 0.55
ADORA2A P29274 2/20 0.55
ADORA2B P29275 2/20 0.55
ADORA1 P30542 2/20 0.55
MEN1 O00255 1/20 0.55
CYP1A2 P05177 1/20 0.55
MAPK1 P28482 1/20 0.55
KMT2A Q03164 1/20 0.55
RXFP1 Q9HBX9 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL26487693 0.90 ADORA3 (0.64) ADORA3ADORA2AADORA2BADORA1MEN1
SCHEMBL28740326 0.89 NT5E (0.72) NT5EADORA3ADORA2AADORA2BADORA1
SCHEMBL26487692 0.88 ADORA3 (0.60) NT5EADORA3ADORA2AADORA2BADORA1
SCHEMBL28740143 0.87 NT5E (0.57) NT5EADORA3ADORA2AADORA2BADORA1
SCHEMBL28740105 0.87 NT5E (0.75) NT5EADORA3ADORA2AADORA2BADORA1
SCHEMBL28740041 0.85 NT5E (0.72) NT5EADORA3ADORA2AADORA2BADORA1
SCHEMBL19100517 0.84 NT5E (0.83) NT5E
SCHEMBL28740153 0.84 NT5E (0.57) NT5EADORA3ADORA2AADORA2BADORA1
SCHEMBL19799156 0.83 ADORA3 (0.79) ADORA3ADORA2AADORA2BADORA1MEN1
SCHEMBL12192981 0.83 ADORA3 (0.79) ADORA3ADORA2AADORA2BADORA1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114395005-A Modulators of extracellular 5' -nucleotidase and uses thereof 艾库斯生物科学有限公司 2022-04-26 CN disclosed