SCHEMBL28746471

SCHEMBL28746471

CCOC(=O)c1[nH]c2ccc(N)cc2c1N

nearest known ligand 0.82

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 10/20 0.82
ALDH1A1 P00352 8/20 0.82
GAA P10253 4/20 0.82
MAPT P10636 3/20 0.82
RAB9A P51151 3/20 0.82
NPC1 O15118 2/20 0.82
SMN1; SMN2 Q16637 2/20 0.82
TP53 P04637 1/20 0.82
HPGD P15428 6/20 0.67
NPSR1 Q6W5P4 1/20 0.67
HTR6 P50406 1/20 0.54
CYP1A2 P05177 2/20 0.50
XBP1 P17861 1/20 0.50
CYP2C19 P33261 1/20 0.50
HSD17B10 Q99714 3/20 0.49
LMNA P02545 2/20 0.49
HTT P42858 1/20 0.49
HCRTR1 O43613 2/20 0.49
CYP3A4 P08684 1/20 0.49
MAOA P21397 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16732481 0.88 KDM4E (0.71) KDM4EALDH1A1GAAMAPTRAB9A
SCHEMBL13758172 0.87 ALDH1A1 (0.76) KDM4EALDH1A1GAAMAPTRAB9A
SCHEMBL31682820 0.87 ALDH1A1 (0.76) KDM4EALDH1A1GAAMAPTRAB9A
SCHEMBL14174305 0.87 ALDH1A1 (0.76) KDM4EALDH1A1GAAMAPTRAB9A
SCHEMBL16747008 0.86 ALDH1A1 (0.61) KDM4EALDH1A1GAAMAPTRAB9A
SCHEMBL1259124 0.86 KDM4E (0.61) KDM4EALDH1A1GAAMAPTRAB9A
Hydrochloric Acid SCHEMBL16732975 0.85 ALDH1A1 (0.60) KDM4EALDH1A1GAAMAPTRAB9A
SCHEMBL4332747 0.84 KDM4E (0.70) KDM4EALDH1A1GAAMAPTRAB9A
SCHEMBL6923876 0.83 KDM4E (0.69) KDM4EALDH1A1GAAMAPTRAB9A
Hydrochloric Acid SCHEMBL8801503 0.82 KDM4E (0.68) KDM4EALDH1A1GAAMAPTRAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114539158-B FXIa inhibitor compound and preparation method and application thereof 沈阳药科大学 2023-12-08 CN disclosed
CN-114539158-A FXIa inhibitor compound and preparation method and application thereof 沈阳药科大学 2022-05-27 CN disclosed