SCHEMBL28751992

SCHEMBL28751992

COc1cc(C(N)=O)cc(N)c1NC/C=C/COC(N)=O

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 1/20 0.39
GAA P10253 2/20 0.38
HTT P42858 2/20 0.37
TSHR P16473 2/20 0.37
APOBEC3A P31941 1/20 0.37
APOBEC3G Q9HC16 1/20 0.37
BPTF Q12830 1/20 0.36
ALDH1A1 P00352 3/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
KDM4E B2RXH2 2/20 0.35
LMNA P02545 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
NCOA1 Q15788 1/20 0.34
NCOA3 Q9Y6Q9 1/20 0.34
CYP1A2 P05177 1/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2C9 P11712 1/20 0.33
CYP2C19 P33261 1/20 0.33
MEN1 O00255 1/20 0.33
HPGD P15428 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22288356 1.00 MAPK1 (0.39) MAPK1GAAHTTTSHRAPOBEC3A
SCHEMBL19451673 0.91 HTT (0.43) MAPK1GAAHTTTSHRAPOBEC3A
SCHEMBL29012732 0.87 HTT (0.33) MAPK1GAAHTTTSHRAPOBEC3A
SCHEMBL23137476 0.86 HTT (0.40) MAPK1GAAHTTTSHRAPOBEC3A
SCHEMBL22150386 0.86 HTT (0.40) MAPK1GAAHTTTSHRAPOBEC3A
SCHEMBL29105274 0.86 ALDH1A1 (0.40) HTTALDH1A1SMN1; SMN2KDM4EMEN1
SCHEMBL29105277 0.86 ALDH1A1 (0.40) HTTALDH1A1SMN1; SMN2KDM4EMEN1
SCHEMBL29868210 0.85 TSHR (0.40) MAPK1HTTTSHRAPOBEC3AAPOBEC3G
SCHEMBL19437548 0.84 HTT (0.38) MAPK1GAAHTTTSHRAPOBEC3A
SCHEMBL19437549 0.84 HTT (0.38) MAPK1GAAHTTTSHRAPOBEC3A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111417630-B Modulators of interferon gene stimulating factor (STING) 葛兰素史克知识产权开发有限公司 2023-06-06 CN disclosed
CN-114585623-A Bis [ N- ((5-carbamoyl) -1H-benzo [ d ] imidazol-2-yl) pyrazole-5-carboxamide ] derivatives and related compounds as STING (interferon gene stimulator) agonists for the treatment of cancer 梅尔莎纳医疗公司 2022-06-03 CN disclosed
CN-111417630-A Modulators of interferon gene stimulating factor (STING) 葛兰素史克知识产权开发有限公司 2020-07-14 CN disclosed