SCHEMBL28752168

SCHEMBL28752168

NC(=O)CC[C@@H]1CN(c2ccc(-c3ccc(C4=NOC(CO)C4)s3)cn2)C(=O)O1

nearest known ligand 0.37

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CETP P11597 1/20 0.36
KCNH2 Q12809 1/20 0.36
NPC1 O15118 1/20 0.36
RAB9A P51151 1/20 0.36
GRM5 P41594 3/20 0.33
F10 P00742 2/20 0.33
ITGB3 P05106 2/20 0.33
ITGA2B P08514 2/20 0.33
CALML3 P27482 3/20 0.31
MAOA P21397 2/20 0.31
MAOB P27338 2/20 0.31
CYP2C19 P33261 2/20 0.30
CYP2C9 P11712 1/20 0.30
MIF P14174 1/20 0.30
CYP3A4 P08684 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3328408 0.84 CETP (0.44) CETPKCNH2F10CALML3MAOA
SCHEMBL13298961 0.84 CETP (0.44) CETPKCNH2F10CALML3MAOA
SCHEMBL4948976 0.81 MAOA (0.49) MAOAMAOBCYP2C9CYP3A4
SCHEMBL3325901 0.79 MAOA (0.42) CETPKCNH2GRM5MAOAMAOB
SCHEMBL3327665 0.73 MAOA (0.48) F10CALML3MAOAMAOB
SCHEMBL3325938 0.70 MAOA (0.52) KCNH2MAOAMAOBCYP2C9CYP3A4
SCHEMBL3068397 0.69 CALML3 (0.54) CALML3MAOAMAOBCYP2C19CYP2C9
SCHEMBL3068395 0.69 CALML3 (0.54) CALML3MAOAMAOBCYP2C19CYP2C9
SCHEMBL3323576 0.69 MAOA (0.49) KCNH2CALML3MAOAMAOB
SCHEMBL3323488 0.69 CALML3 (0.60) F10CALML3MAOAMAOBCYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1639136-A Oxazolidinone and/or isoxazoline as antibacterial agents ASTRAZENECA AB (SE) 2005-07-13 CN disclosed