Hydantoin

Hydantoin

SCHEMBL2875362

CC(=O)O.O=C1CNC(=O)N1

nearest known ligand 0.46

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ADRA2AADRA2BADRA2CADRB2AGTR1AVPR1AAVPR1BAVPR2BDKRB2CALCRCHRNA3CHRNB4ESR1ESR2GHSRGNRHRGSC1HSPA8MALT1MC1RMC4RNOS1NOS2NOS3OPRK1OXTRRAMP1RAMP2RAMP3SCN5ASSTR1SSTR2SSTR3SSTR4SSTR5dacAdacBdacCfolPftsImrcAmrcBmrdArplArplBrplCrplDrplErplFrplJrplKrplLrplMrplNrplOrplPrplQrplRrplSrplTrplUrplVrplWrplXrplYrpmArpmBrpmCrpmDrpmErpmFrpmGrpmHrpmIrpmJrpsArpsBrpsCrpsDrpsErpsFrpsGrpsHrpsIrpsJrpsKrpsLrpsMrpsNrpsOrpsPrpsQrpsRrpsSrpsTrpsUykgMykgO

The experimentally established mechanism targets of Hydantoin. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CRBN Q96SW2 2/20 0.41
MB P02144 2/20 0.34
FFAR3 O14843 1/20 0.33
LCK P06239 1/20 0.33
FYN P06241 1/20 0.33
ITGB3 P05106 1/20 0.32
ITGB1 P05556 1/20 0.32
ITGAV P06756 1/20 0.32
ITGA4 P13612 1/20 0.32
PDE3B Q13370 1/20 0.31
PDE3A Q14432 1/20 0.31
USP2 O75604 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydantoin SCHEMBL10636755 0.93 CRBN (0.42) CRBNMBPDE3BPDE3A
Hydantoin SCHEMBL28140889 0.90 CRBN (0.44) CRBNMBITGB3ITGB1ITGAV
Hydantoin SCHEMBL11127367 0.86 CRBN (0.41) CRBNMBPDE3BPDE3A
Hydantoin SCHEMBL27705088 0.84 CRBN (0.52) CRBNMBPDE3BPDE3A
Hydantoin SCHEMBL27690 0.84
Hydantoin SCHEMBL7285865 0.84
Hydantoin SCHEMBL28531040 0.84 CRBN (0.33) CRBN
Hydantoin SCHEMBL27655704 0.84 CRBN (0.39) CRBNMBITGB3ITGB1ITGAV
Hydantoin SCHEMBL16971290 0.83 CRBN (0.42) CRBNMB
Hydantoin SCHEMBL27574136 0.82 CRBN (0.46) CRBNMBPDE3BPDE3A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 25 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5939556-A Hydantoin compounds, salts thereof, processes for their preparation, and processes for preparing pharmaceutically active compounds comprising them HOECHST AKTIENGESELLSCHAFT (DE) 1999-08-17 US claimed
EP-0628571-A1 NOVEL PEPTIDE, AND ANTITHROMBOTIC AGENT, ANTICOAGULANT FOR EXTRACORPOREAL CIRCULATION, CELL FUSION INHIBITOR, CANCER METASTASIS INHIBITOR, PROTECTIVE FOR PLATELET PREPARATION FOR TRANSFUSION AND PACK OF PLATELET PREPARATION FOR TRANSFUSION NIPPON STEEL CORPORATION (JP) 1994-12-14 EP claimed
EP-0422765-A1 Cosmetic composition UNILEVER PLC (GB) 1991-04-17 EP claimed
CN-109153644-B Small molecules against CEREBLON to enhance effector T cell function H·李·莫菲特癌症中心研究有限公司 2022-10-21 CN disclosed
CN-101379138-B Conductive polymer solution, conductive coating film, capacitor and method for producing same 信越聚合物株式会社 2019-03-22 CN disclosed
CN-109153644-A SMALL MOLECULES AGAINST CEREBLON TO ENHANCE EFFECTOR T CELL FUNCTION H·李·莫菲特癌症中心研究有限公司 2019-01-04 CN disclosed
CN-104496912-A Preparation method for orotic acid INST SUBTROPICAL AGRI CAS 2015-04-08 CN disclosed
US-7662845-B2 2,5-Dioxoimidazolidin-4-yl acetamides and analogues as inhibitors of metalloproteinase MMP12 ASTRAZENECA AB (SE) 2010-02-16 US disclosed
CN-100398521-C 2,5-dioxoimidazolidin-4-yl acetamides and analogues as inhibitors of metalloproteinase MMP12 ASTRAZENECA AB (SE) 2008-07-02 CN disclosed
US-7354940-B2 2,5-dioxoimidazolidin-4-yl acetamines and analogues as inhibitors of metalloproteinase mmp12 ASTRAZENECA AB (SE) 2008-04-08 US disclosed
EP-1542977-B1 2,5-DIOXOIMIDAZOLIDIN-4-YL ACETAMIDES AND ANALOGUES AS INHIBITORS OF METALLOPROTEINASE MMP12. ASTRAZENECA AB (SE) 2006-12-20 EP disclosed
CN-1125054-C Novel imidazolidine derivatives, their preparation, their use and pharmaceutical preparations comprising them AVENTIS PHARMACEUTICS GMBH (DE) 2003-10-22 CN disclosed
CN-1267210-A Hair styling composition PROCTER & GAMBLE (US) 2000-09-20 CN disclosed
US-5939556-A Hydantoin compounds, salts thereof, processes for their preparation, and processes for preparing pharmaceutically active compounds comprising them HOECHST AKTIENGESELLSCHAFT (DE) 1999-08-17 US disclosed
CN-1218047-A Novel imidazolidine derivatives, their preparation, their use and pharmaceutical preparations comprising them HOECHST MARION ROUSSEL DE GMBH (DE) 1999-06-02 CN disclosed
CN-1037975-C Curable suspensions of epoxy resins CIBA GEIGY AG (CH) 1998-04-08 CN disclosed
US-5498601-A RGD SEQUENCE NIPPON STEEL CORPORATION (JP) 1996-03-12 US disclosed
EP-0628571-A1 NOVEL PEPTIDE, AND ANTITHROMBOTIC AGENT, ANTICOAGULANT FOR EXTRACORPOREAL CIRCULATION, CELL FUSION INHIBITOR, CANCER METASTASIS INHIBITOR, PROTECTIVE FOR PLATELET PREPARATION FOR TRANSFUSION AND PACK OF PLATELET PREPARATION FOR TRANSFUSION NIPPON STEEL CORPORATION (JP) 1994-12-14 EP disclosed
CN-1083082-A Curable suspensions of epoxy resins CIBA GEIGY AG (CH) 1994-03-02 CN disclosed
EP-0422765-A1 Cosmetic composition UNILEVER PLC (GB) 1991-04-17 EP disclosed