SCHEMBL28756490

SCHEMBL28756490

COc1cc2ncc(C#N)c(Nc3ccccc3)c2cc1OC

nearest known ligand 0.95

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
MAP2K1 Q02750 7/20 0.95
RAF1 P04049 2/20 0.83
EGFR P00533 12/20 0.80
ERBB2 P04626 11/20 0.80
SRC P12931 2/20 0.78
GAK O14976 2/20 0.77

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6382750 0.91 MAP2K1 (1.00) MAP2K1RAF1EGFRERBB2SRC
SCHEMBL6384880 0.89 MAP2K1 (1.00) MAP2K1RAF1EGFRERBB2SRC
SCHEMBL6381609 0.89 EGFR (1.00) MAP2K1RAF1EGFRERBB2SRC
SCHEMBL6381535 0.88 EGFR (1.00) MAP2K1RAF1EGFRERBB2SRC
SCHEMBL6381446 0.88 EGFR (1.00) MAP2K1RAF1EGFRERBB2SRC
SCHEMBL6381926 0.88 MAP2K1 (0.76) MAP2K1EGFRERBB2SRCGAK
SCHEMBL6383704 0.88 EGFR (0.78) MAP2K1RAF1EGFRERBB2SRC
SCHEMBL5733290 0.88 MAP2K1 (1.00) MAP2K1RAF1EGFRERBB2SRC
SCHEMBL6381464 0.88 EGFR (1.00) MAP2K1RAF1EGFRERBB2SRC
SCHEMBL6380423 0.88 EGFR (1.00) MAP2K1EGFRERBB2SRCGAK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-100432071-C Substituted 1H-indole-2-ketone compound and its preparation method and uses SHANGHAI INST MATERIA MEDICA (CN) 2008-11-12 CN disclosed
CN-1769284-A Substituted 1H-indole-2-ketone compound and its preparation method and uses SHANGHAI INST MATERIA MEDICA (CN) 2006-05-10 CN disclosed