SCHEMBL28757646

SCHEMBL28757646

FC(F)(F)c1cccc(-c2ccc3c(Nc4ccc(C(Cl)(Cl)Cl)cc4)nncc3c2)n1

nearest known ligand 0.41

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
EGFR P00533 6/20 0.41
KDR P35968 6/20 0.41
EPHX2 P34913 5/20 0.37
CA9 Q16790 1/20 0.36
ACP1 P24666 1/20 0.35
PIM1 P11309 1/20 0.35
PIM3 Q86V86 1/20 0.35
PIM2 Q9P1W9 1/20 0.35
MEN1 O00255 1/20 0.35
RAB9A P51151 1/20 0.35
KMT2A Q03164 1/20 0.35
CTDSP1 Q9GZU7 1/20 0.35
TDP1 Q9NUW8 1/20 0.35
TRPV1 Q8NER1 1/20 0.35
NOTUM Q6P988 1/20 0.34
TGFBR1 P36897 2/20 0.34
TGFBR2 P37173 1/20 0.33
BRAF P15056 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4678972 0.93 EGFR (0.43) EGFRKDREPHX2CA9ACP1
SCHEMBL4674839 0.79 TRPV1 (0.47) EGFRKDREPHX2ACP1MEN1
SCHEMBL4675893 0.77 KIF11 (0.44) EGFRKDREPHX2ACP1MEN1
SCHEMBL4674553 0.75 EPHX2 (0.42) EGFRKDREPHX2ACP1MEN1
SCHEMBL4675714 0.73 EPHX2 (0.62) EGFRKDREPHX2ACP1MEN1
SCHEMBL4678999 0.72 TRPV1 (0.47) EGFRKDRMEN1KMT2ATRPV1
SCHEMBL27657900 0.72 EPHX2 (0.37) EGFRKDREPHX2CA9TRPV1
SCHEMBL4677054 0.71 EGFR (0.43) EGFRKDREPHX2ACP1MEN1
SCHEMBL4675491 0.71 EPHX2 (0.53) EGFRKDREPHX2ACP1MEN1
SCHEMBL4674768 0.71 TRPV1 (0.47) EGFRKDREPHX2ACP1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1816541-A Substituted-1-phthalazinamines as vr-1 antagonists MERCK SHARP & DOHME (GB) 2006-08-09 CN disclosed