SCHEMBL28758201

SCHEMBL28758201

CC(C=O)c1cc(Cl)ccc1OC(F)(F)F

nearest known ligand 0.37

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
APP P05067 1/20 0.37
CNR2 P34972 2/20 0.36
CYP11B1 P15538 1/20 0.36
CYP11B2 P19099 1/20 0.36
ANO1 Q5XXA6 2/20 0.35
ALPL P05186 4/20 0.34
TNNI3K Q59H18 2/20 0.34
F11 P03951 1/20 0.34
HTR2A P28223 2/20 0.34
TSHR P16473 1/20 0.34
HTR2C P28335 1/20 0.34
HTR2B P41595 1/20 0.34
PNLIP P16233 1/20 0.34
SLC6A4 P31645 2/20 0.33
KCNH2 Q12809 1/20 0.33
FFAR4 Q5NUL3 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12356955 0.82 KCNK3 (0.39) APPCNR2ALPLF11HTR2A
SCHEMBL28755485 0.82 HRH4 (0.37) APPALPLSLC6A4
SCHEMBL6445833 0.82 EPAS1 (0.34) APPCNR2CYP11B1CYP11B2ANO1
SCHEMBL16957725 0.80 CNR2 (0.35) APPCNR2ANO1ALPLF11
SCHEMBL20303532 0.80 PDE2A (0.42) APPCNR2ANO1ALPLF11
SCHEMBL19262097 0.80 CNR2 (0.38) APPCNR2ANO1ALPLF11
SCHEMBL27643654 0.78 ANO1 (0.34) APPCNR2CYP11B1CYP11B2ANO1
SCHEMBL27624241 0.78 KCNK3 (0.44) APPCYP11B1CYP11B2SLC6A4KCNH2
SCHEMBL32682742 0.75 CNR2 (0.40) CNR2ALPLTNNI3KF11
SCHEMBL20303378 0.75 CNR2 (0.40) CNR2ALPLTNNI3KF11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-100395234-C Novel CB1 receptor inverse agonists HOFFMANN LA ROCHE (CH) 2008-06-18 CN disclosed
CN-101012193-A Novel CB 1 receptour inverse agonists HOFFMANN LA ROCHE (CH) 2007-08-08 CN disclosed
CN-1735593-A Novel CB1 receptor inverse agonists HOFFMANN LA ROCHE (CH) 2006-02-15 CN disclosed