SCHEMBL28759591

SCHEMBL28759591

C[N+](C)(C)Nc1nc(N)nc2cc(-c3ccccc3C(F)(F)F)c3[nH]ccc3c12

nearest known ligand 0.40

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
PTPN1 P18031 8/20 0.40
C1R P00736 1/20 0.35
CYP1A2 P05177 1/20 0.34
CYP2D6 P10635 1/20 0.34
CYP2C19 P33261 1/20 0.34
RECQL P46063 1/20 0.34
DHFR P00374 2/20 0.34
TRPA1 O75762 3/20 0.33
BACE1 P56817 1/20 0.33
TRPM8 Q7Z2W7 1/20 0.32
TRPV1 Q8NER1 1/20 0.32
TTBK1 Q5TCY1 1/20 0.32
TTBK2 Q6IQ55 1/20 0.32
ULK1 O75385 1/20 0.32
ACP1 P24666 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4691348 0.83 DHFR (0.41) PTPN1C1RDHFRTRPA1BACE1
SCHEMBL27653772 0.83 TTBK1 (0.39) DHFRTTBK1TTBK2
SCHEMBL27653789 0.81 CYP1A2 (0.43) PTPN1C1RCYP1A2CYP2D6CYP2C19
SCHEMBL27633378 0.77 PTPN1 (0.36) PTPN1C1RCYP1A2CYP2D6DHFR
SCHEMBL28759599 0.77 DHFR (0.34) DHFR
SCHEMBL27653795 0.75 DHFR (0.32) DHFR
SCHEMBL4689031 0.69 DHFR (0.58) DHFR
SCHEMBL27653903 0.69 DHFR (0.38) DHFRTTBK1TTBK2
SCHEMBL4691907 0.69 DHFR (0.43) PTPN1C1RDHFRTRPA1BACE1
SCHEMBL4707590 0.68 PTPN1 (0.48) PTPN1CYP1A2CYP2D6CYP2C19RECQL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-100334088-C Diaminopyrroloquinazoline compounds as protein tyrosine phosphatase inhibitors HOFFMANN LA ROCHE CO LTD (CH) 2007-08-29 CN disclosed
CN-1791604-A Diaminopyrroloquinazolines compounds as protein tyrosine phosphatase inhibitors HOFFMANN LA ROCHE (CH) 2006-06-21 CN disclosed