SCHEMBL28759740

SCHEMBL28759740

CS(=O)(=O)OCc1cc2c(cn1)CCN(C(=O)O)C2

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 0.35
NPC1 O15118 1/20 0.35
GPR183 P32249 1/20 0.34
HRH3 Q9Y5N1 1/20 0.34
MEN1 O00255 2/20 0.34
ALDH1A1 P00352 2/20 0.33
STS P08842 2/20 0.33
KDM4E B2RXH2 1/20 0.33
TSHR P16473 1/20 0.33
HSD17B10 Q99714 1/20 0.33
ESR1 P03372 1/20 0.33
CA1 P00915 1/20 0.33
CA2 P00918 1/20 0.33
CA7 P43166 1/20 0.33
CA9 Q16790 1/20 0.33
CA14 Q9ULX7 1/20 0.33
HPGD P15428 1/20 0.33
TMEM97 Q5BJF2 1/20 0.33
SIGMAR1 Q99720 1/20 0.33
HDAC1 Q13547 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29723003 0.85 ESR2 (0.51) MAPK1
SCHEMBL21591662 0.85 HDAC1 (0.43) KMT2ANPC1GPR183MEN1ALDH1A1
SCHEMBL23301570 0.81 ESR2 (0.54) MAPK1
SCHEMBL29712337 0.81 ESR2 (0.54) MAPK1
SCHEMBL29077472 0.78 KMT2A (0.34) KMT2ANPC1GPR183MEN1KDM4E
SCHEMBL28675076 0.78 TMEM97 (0.43) KMT2ANPC1GPR183HRH3ALDH1A1
SCHEMBL6282952 0.78 HSP90AA1 (0.40) HSP90AA1HSP90B1
SCHEMBL17242052 0.76 USP30 (0.36)
SCHEMBL29155326 0.76 ESR2 (0.43) KMT2ANPC1GPR183ALDH1A1HSD17B10
SCHEMBL3441436 0.72 HDAC6 (0.39) KMT2ANPC1ALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114621230-B Nitrogen-containing heterocyclic compound, preparation method thereof and application thereof in medicine 江苏恒瑞医药股份有限公司 2023-06-16 CN disclosed
CN-114621230-A Nitrogen-containing heterocyclic compound, preparation method and medical application thereof 江苏恒瑞医药股份有限公司 2022-06-14 CN disclosed