SCHEMBL28759793

SCHEMBL28759793

COc1cc2ncnc(Oc3ccc(C(F)(F)C(=O)Nc4cc(C(F)(F)F)cc(C(F)(F)F)c4)cc3)c2cc1OC

nearest known ligand 0.73

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
KDR P35968 12/20 0.73
BRAF P15056 10/20 0.70
MAPK14 Q16539 2/20 0.70
TNNI3K Q59H18 2/20 0.70
RAF1 P04049 5/20 0.65
PDGFRA P16234 1/20 0.60
CSF1R P07333 1/20 0.58
EGFR P00533 1/20 0.56
FGFR4 P22455 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28759802 0.95 BRAF (0.72) KDRBRAFMAPK14TNNI3KRAF1
SCHEMBL29723022 0.95 BRAF (0.72) KDRBRAFMAPK14TNNI3KRAF1
SCHEMBL29723231 0.93 BRAF (0.82) KDRBRAFMAPK14TNNI3KRAF1
SCHEMBL28759820 0.93 BRAF (0.82) KDRBRAFMAPK14TNNI3KRAF1
SCHEMBL28759806 0.89 KDR (0.73) KDRBRAFMAPK14TNNI3KRAF1
SCHEMBL29722991 0.89 KDR (0.73) KDRBRAFMAPK14TNNI3KRAF1
SCHEMBL29722983 0.87 KDR (0.67) KDRBRAFMAPK14TNNI3KRAF1
SCHEMBL28759810 0.87 KDR (0.67) KDRBRAFMAPK14TNNI3KRAF1
SCHEMBL30447746 0.86 KDR (0.69) KDRBRAFMAPK14TNNI3KRAF1
SCHEMBL28759809 0.86 BRAF (0.72) KDRBRAFMAPK14TNNI3KRAF1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114621140-B Aryldifluoroacetamide compound, preparation method and application thereof 中国科学院上海药物研究所 2023-08-11 CN disclosed
CN-114621140-A Aryl difluoro acetamide compound and preparation method and application thereof 中国科学院上海药物研究所 2022-06-14 CN disclosed