SCHEMBL28760141

SCHEMBL28760141

NC(=O)N(c1ccccc1)c1ccc(-c2ccc(F)c3[nH]nc(N)c23)cc1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDR P35968 13/20 0.57
FLT3 P36888 10/20 0.52
KIT P10721 9/20 0.52
CSF1R P07333 6/20 0.42
FLT1 P17948 5/20 0.42
MET P08581 5/20 0.42
PRKACA P17612 5/20 0.42
ROCK1 Q13464 5/20 0.42
FLT4 P35916 5/20 0.42
LCK P06239 4/20 0.42
GSK3A P49840 4/20 0.42
CDK5 Q00535 4/20 0.42
DYRK1A Q13627 4/20 0.42
NTRK1 P04629 4/20 0.42
FGFR1 P11362 4/20 0.42
LYN P07948 4/20 0.42
PLK4 O00444 4/20 0.42
AURKA O14965 4/20 0.42
ROCK2 O75116 4/20 0.42
CDK1 P06493 4/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27636388 0.92 KDR (0.56) KDRFLT3KITCSF1RFLT1
SCHEMBL27657327 0.90 KDR (0.62) KDRFLT3KITCSF1RFLT1
SCHEMBL27657458 0.90 KDR (0.57) KDRFLT3KITCSF1RFLT1
SCHEMBL27657350 0.89 KDR (0.56) KDRFLT3KITCSF1RFLT1
SCHEMBL27636555 0.87 KDR (0.48) KDRFLT3KITCSF1RFLT1
SCHEMBL27657341 0.87 KDR (0.54) KDRFLT3KITCSF1RFLT1
SCHEMBL27657333 0.87 KDR (0.54) KDRFLT3KITCSF1RFLT1
SCHEMBL27657282 0.86 KDR (0.54) KDRFLT3KITCSF1RFLT1
SCHEMBL27657312 0.84 KDR (0.52) KDRFLT3KITCSF1RFLT1
SCHEMBL27657352 0.82 KDR (0.66) KDRFLT3KITCSF1RFLT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1826324-B indazole, Benzisoxazole and benzisothiazole kinase inhibitors ABBOTT LABORATORIES (US) 2011-12-07 CN claimed
CN-1826324-A Indazole, benzisoxazole and benzisothiazole kinase inhibitors ABBOTT LAB (US) 2006-08-30 CN claimed
CN-102417487-A Indazole, benzisoxazole and benzisothiazole kinase inhibitors ABBOTT LAB 2012-04-18 CN disclosed
CN-1826324-B indazole, Benzisoxazole and benzisothiazole kinase inhibitors ABBOTT LABORATORIES (US) 2011-12-07 CN disclosed
CN-101827584-A Solid dispersion product of N-aryl ureido drugs ABBOTT GMBH & CO KG 2010-09-08 CN disclosed
CN-1826324-A Indazole, benzisoxazole and benzisothiazole kinase inhibitors ABBOTT LAB (US) 2006-08-30 CN disclosed