SCHEMBL28760185

SCHEMBL28760185

c1ccc(C(c2ccccc2)N2CCN(Cc3cccnc3)CC2)cc1

nearest known ligand 0.63

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ATM Q13315 2/20 0.63
CHRNB2 P17787 1/20 0.60
CHRNA4 P43681 1/20 0.60
TRPV6 Q9H1D0 2/20 0.56
OPRD1 P41143 1/20 0.56
ALDH1A1 P00352 3/20 0.54
KDM4E B2RXH2 2/20 0.54
TDP1 Q9NUW8 1/20 0.54
TP53 P04637 1/20 0.54
MEN1 O00255 1/20 0.53
KMT2A Q03164 1/20 0.53
USP2 O75604 1/20 0.52
CYP1A2 P05177 1/20 0.52
CYP3A4 P08684 1/20 0.52
CYP2D6 P10635 1/20 0.52
CYP2C19 P33261 1/20 0.52
HPN P05981 1/20 0.52
CHRM2 P08172 1/20 0.52
ADRA2A P08913 1/20 0.52
ADORA3 P0DMS8 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7311276 0.85 ATM (0.84) ATMOPRD1KDM4EMEN1KMT2A
SCHEMBL15800693 0.85 CHRNB2 (0.77) CHRNB2CHRNA4TRPV6ALDH1A1KDM4E
Hydrochloric Acid SCHEMBL16226937 0.83 ATM (0.82) ATMOPRD1KDM4EMEN1KMT2A
SCHEMBL16026435 0.83 CHRNB2 (0.85) CHRNB2CHRNA4TRPV6ALDH1A1KDM4E
SCHEMBL30122798 0.81 CHRNB2 (0.66) CHRNB2CHRNA4TRPV6ALDH1A1KDM4E
SCHEMBL13412386 0.81 CHRNB2 (0.66) CHRNB2CHRNA4TRPV6ALDH1A1KDM4E
SCHEMBL4474652 0.81 KDM4E (0.74) CHRNB2CHRNA4TRPV6OPRD1ALDH1A1
SCHEMBL20804485 0.80 CHRNB2 (0.53) CHRNB2CHRNA4TRPV6ALDH1A1KDM4E
SCHEMBL31350803 0.80 CYP3A4 (0.61) ATMOPRD1ALDH1A1MEN1KMT2A
Ammonia Solution, Strong SCHEMBL20740614 0.79 CHRNB2 (0.64) CHRNB2CHRNA4TRPV6ALDH1A1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-100502868-C 3CL protease inhibitor of non-peptide SARS coronavirus and use thereof UNIV BEIJING (CN) 2009-06-24 CN claimed
CN-1965833-A 3CL protease inhibitor of non-peptide SARS coronavirus and use thereof UNIV BEIJING (CN) 2007-05-23 CN claimed
CN-100502868-C 3CL protease inhibitor of non-peptide SARS coronavirus and use thereof UNIV BEIJING (CN) 2009-06-24 CN disclosed
CN-1965833-A 3CL protease inhibitor of non-peptide SARS coronavirus and use thereof UNIV BEIJING (CN) 2007-05-23 CN disclosed