SCHEMBL28761672

SCHEMBL28761672

CN(C=O)c1cc2ncccc2[nH]1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ATAD2 Q6PL18 1/20 0.50
MAPT P10636 2/20 0.47
SNCA P37840 1/20 0.47
DAO P14920 1/20 0.46
HRH4 Q9H3N8 1/20 0.40
CNR2 P34972 1/20 0.35
AURKA O14965 2/20 0.34
KCNMA1 Q12791 1/20 0.34
DRD3 P35462 1/20 0.34
NPC1 O15118 1/20 0.32
GAA P10253 1/20 0.32
RAB9A P51151 1/20 0.32
FGFR1 P11362 1/20 0.32
KDM4E B2RXH2 1/20 0.32
NPSR1 Q6W5P4 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
PTGDR2 Q9Y5Y4 1/20 0.31
CDK1 P06493 1/20 0.31
CDK2 P24941 1/20 0.31
MKNK1 Q9BUB5 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25775091 0.82 MAPT (0.56) ATAD2MAPTSNCADAOHRH4
SCHEMBL29422812 0.71 DAO (0.53) ATAD2MAPTSNCADAOHRH4
SCHEMBL4278906 0.71 DAO (0.53) ATAD2MAPTSNCADAOHRH4
SCHEMBL24449652 0.70 ATAD2 (0.44) ATAD2MAPTSNCADAOHRH4
SCHEMBL4641753 0.69 ATAD2 (0.62) ATAD2MAPTSNCADAOHRH4
SCHEMBL29997480 0.69 ATAD2 (0.62) ATAD2MAPTSNCADAOHRH4
SCHEMBL9396747 0.68 ATAD2 (0.49) ATAD2MAPTSNCADAOHRH4
SCHEMBL17480050 0.68 DOT1L (0.54) MAPTNPC1RAB9AKDM4ESMN1; SMN2
SCHEMBL18590950 0.67 ATAD2 (0.42) ATAD2MAPTSNCADAOHRH4
SCHEMBL30663285 0.67 ATAD2 (1.00) ATAD2MAPTSNCADAOHRH4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-100439367-C Substituted 1H-pyrrolo[3,2-b, 3,2-c, and 2,3-c]pyridine-2-carboxamides and related analogs as inhibitors of casein kinase lepsilon AVENTIS PHARMA INC (US) 2008-12-03 CN disclosed
CN-1906194-A Substituted 1H-pyrrolo [3, 2-b, 3, 2-c and 2, 3-c ] pyridine-2-carboxamides and related analogs as inhibitors of casein kinase ie AVENTIS PHARMA INC (US) 2007-01-31 CN disclosed