SCHEMBL28763538

SCHEMBL28763538

[CH2]c1ccc(-c2scnc2C)cc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
VHL P40337 11/20 0.50
PDE10A Q9Y233 2/20 0.35
KDM4E B2RXH2 3/20 0.34
PKM P14618 1/20 0.34
ELOC Q15369 2/20 0.33
ELOB Q15370 2/20 0.33
MEN1 O00255 1/20 0.33
ALDH1A1 P00352 1/20 0.33
LMNA P02545 1/20 0.33
CYP1A2 P05177 1/20 0.33
CYP2D6 P10635 1/20 0.33
CYP2C9 P11712 1/20 0.33
CYP2C19 P33261 1/20 0.33
KMT2A Q03164 1/20 0.33
PDE4D Q08499 1/20 0.31
PDE3A Q14432 1/20 0.31
P2RX3 P56373 1/20 0.31
P2RX2 Q9UBL9 1/20 0.31
CYP4F2 P78329 1/20 0.31
CYP4A11 Q02928 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19661678 0.83 VHL (0.53) VHLKDM4EPKMELOCELOB
SCHEMBL18579787 0.83 VHL (0.57) VHLKDM4EELOCELOBMEN1
SCHEMBL19600685 0.80 VHL (0.54) VHLKDM4EPKMELOCELOB
SCHEMBL22130274 0.80 VHL (0.50) VHLKDM4EPKMELOCELOB
SCHEMBL25006423 0.79 VHL (0.47) VHLPDE10AKDM4EPKMELOC
SCHEMBL679793 0.79 KDM4E (0.53) VHLKDM4EPKMMEN1ALDH1A1
SCHEMBL16276343 0.77 VHL (0.59) VHLKDM4EELOCELOBMEN1
SCHEMBL16300950 0.77 ALOX5 (0.49) VHLKDM4EMEN1ALDH1A1KMT2A
SCHEMBL17947426 0.77 VHL (0.48) VHLKDM4EALDH1A1P2RX3P2RX2
SCHEMBL23478765 0.77 VHL (0.48) VHLKDM4EELOCELOBALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109678852-B 6-oxo-hexahydropyrimidine derivative, preparation method and pharmaceutical application thereof 南京中医药大学 2022-04-19 CN claimed
CN-109678852-B 6-oxo-hexahydropyrimidine derivative, preparation method and pharmaceutical application thereof 南京中医药大学 2022-04-19 CN disclosed