SCHEMBL28763543

SCHEMBL28763543

Fc1ccc(CCBr)c(C(F)(F)F)c1

nearest known ligand 0.56

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 2/20 0.56
SLC6A2 P23975 8/20 0.40
SLC6A4 P31645 8/20 0.40
HDAC3 O15379 1/20 0.40
HDAC1 Q13547 1/20 0.40
HDAC2 Q92769 1/20 0.40
HDAC6 Q9UBN7 1/20 0.40
P2RX7 Q99572 6/20 0.39
SLC6A3 Q01959 1/20 0.39
DHFR P00374 1/20 0.38
GPR183 P32249 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18007055 0.86 IDO1 (0.50) IDO1SLC6A2SLC6A4HDAC3HDAC1
SCHEMBL488748 0.84 IDO1 (0.59) IDO1SLC6A2SLC6A4HDAC3HDAC1
SCHEMBL29616489 0.84 IDO1 (0.59) IDO1SLC6A2SLC6A4HDAC3HDAC1
SCHEMBL27975927 0.81 DAO (0.51) IDO1SLC6A4
SCHEMBL2296868 0.81 KDM1A (0.41) IDO1SLC6A4GPR183
SCHEMBL7782539 0.81 IDO1 (0.61) IDO1SLC6A2SLC6A4HDAC3HDAC1
SCHEMBL22445529 0.81 IDO1 (0.56) IDO1SLC6A2SLC6A4HDAC3HDAC1
SCHEMBL17071866 0.81 IDO1 (0.56) IDO1SLC6A2SLC6A4HDAC3HDAC1
SCHEMBL1538597 0.79 IDO1 (0.63) IDO1SLC6A2SLC6A4HDAC3HDAC1
SCHEMBL27851289 0.79 POLQ (0.43) IDO1SLC6A4P2RX7GPR183

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103265477-A Aminoheteroaryl compounds as protein kinase inhibitors SUGEN INC 2013-08-28 CN disclosed
CN-101023064-B Enantiomerically pure aminoheteroaryl compounds as protein kinase inhibitors PFIZER 2011-02-16 CN disclosed
CN-101023064-A Enantiomerically pure aminoheteroaryl compounds as protein kinase inhibitors AGOURON PHARMA (US) 2007-08-22 CN disclosed