SCHEMBL28767553

SCHEMBL28767553

O=CCC1CCCc2ccc(Cl)cc21

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4C Q9H3R0 2/20 0.46
HTR2A P28223 5/20 0.43
HTR2C P28335 5/20 0.43
HTR2B P41595 5/20 0.43
ADRB1 P08588 1/20 0.38
HTR1A P08908 1/20 0.38
ADRA2A P08913 1/20 0.38
ADRA2B P18089 1/20 0.38
ADRA2C P18825 1/20 0.38
CNR1 P21554 1/20 0.38
SLC6A2 P23975 1/20 0.38
SLC6A4 P31645 1/20 0.38
HRH1 P35367 1/20 0.38
KCNH2 Q12809 1/20 0.38
DRD2 P14416 1/20 0.38
DRD4 P21917 1/20 0.38
ESR1 P03372 1/20 0.35
ESR2 Q92731 1/20 0.35
TAS1R3 Q7RTX0 1/20 0.35
TAS1R1 Q7RTX1 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29673185 1.00 KDM4C (0.46) KDM4CHTR2AHTR2CHTR2BADRB1
SCHEMBL28766634 0.88 KDM4C (0.46) KDM4CHTR2AHTR2CHTR2BESR1
SCHEMBL13229181 0.82 ACHE (0.38) MEN1KMT2AACHE
Hydrochloric Acid SCHEMBL30299242 0.81 HTR2A (0.46) KDM4CHTR2AHTR2CHTR2BADRB1
SCHEMBL15818869 0.80 HTR2A (0.47) KDM4CHTR2AHTR2CHTR2BADRB1
SCHEMBL5467690 0.78 IDO1 (0.47) KDM4C
SCHEMBL24542989 0.76 HTR2C (0.41) KDM4CHTR2AHTR2CHTR2BADRB1
SCHEMBL29673081 0.76 HTR2C (0.41) KDM4CHTR2AHTR2CHTR2BADRB1
Hydrochloric Acid SCHEMBL1066112 0.74 ACHE (0.48) KDM4CHTR2AHTR2CHTR2BADRB1
Hydrochloric Acid SCHEMBL1002239 0.74 ACHE (0.48) KDM4CHTR2AHTR2CHTR2BADRB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022127827-A1 KRASG12C PROTEIN MUTATION INHIBITOR AND PREPARATION METHOD THEREFOR, PHARMACEUTICAL COMPOSITION AND APPLICATION THEREOF 上海维申医药有限公司 2022-06-23 WO disclosed
CN-114644631-A KRAS G12C protein mutation inhibitor, preparation method thereof, pharmaceutical composition and application thereof 上海维申医药有限公司 2022-06-21 CN disclosed