SCHEMBL28772200

SCHEMBL28772200

N#Cc1ccc(F)c(C(c2cc(N)ncc2Cl)S(=O)(=O)CC=Cc2ccc(Cl)cc2)c1

nearest known ligand 0.33

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
TRPV4 Q9HBA0 1/20 0.33
SCN1A P35498 1/20 0.33
SCN5A Q14524 1/20 0.33
SCN8A Q9UQD0 1/20 0.33
S1PR3 Q99500 4/20 0.33
TNF P01375 1/20 0.31
PSEN1 P49768 1/20 0.31
PSEN2 P49810 1/20 0.31
APH1B Q8WW43 1/20 0.31
NCSTN Q92542 1/20 0.31
APH1A Q96BI3 1/20 0.31
PSENEN Q9NZ42 1/20 0.31
GRIK1 P39086 1/20 0.31
GRIK2 Q13002 1/20 0.31
GRM5 P41594 1/20 0.30
S1PR1 P21453 2/20 0.30
S1PR4 O95977 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1631121 0.81 PSEN1 (0.38) TRPV4SCN1ASCN5ASCN8AS1PR3
SCHEMBL28772202 0.78 S1PR3 (0.36) TRPV4SCN1ASCN5ASCN8AS1PR3
SCHEMBL1632894 0.72 PSEN1 (0.42) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL1631914 0.71 PSEN1 (0.39) TRPV4SCN1ASCN5ASCN8AS1PR3
SCHEMBL12762203 0.68 PSEN1 (0.38) TRPV4SCN1ASCN5ASCN8AS1PR3
SCHEMBL1632260 0.67 PSEN1 (0.53) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL1631232 0.66 SCN1A (0.41) SCN1ASCN5ASCN8AS1PR3TNF
SCHEMBL1632245 0.66 PSEN1 (0.37) SCN1ASCN5ASCN8AS1PR3TNF
SCHEMBL1633173 0.66 PSEN1 (0.40) SCN1ASCN5ASCN8ATNFPSEN1
SCHEMBL1631897 0.64 PSEN1 (0.48) PSEN1PSEN2APH1BNCSTNAPH1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-100378072-C Heterocyclic methyl sulfone derivative DAIICHI SEIYAKU CO (JP) 2008-04-02 CN disclosed