SCHEMBL28772202

SCHEMBL28772202

C=CC(c1ccc(Cl)cc1)S(=O)(=O)C(c1cc(C#N)ccc1F)c1cc(N)ncc1Cl

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
S1PR3 Q99500 10/20 0.36
S1PR1 P21453 5/20 0.34
S1PR4 O95977 1/20 0.34
SCN1A P35498 2/20 0.33
SCN5A Q14524 2/20 0.33
SCN8A Q9UQD0 2/20 0.33
TRPV4 Q9HBA0 1/20 0.32
TNF P01375 1/20 0.31
PIK3CA P42336 1/20 0.31
PIK3CB P42338 1/20 0.31
MTOR P42345 1/20 0.31
PIK3CG P48736 1/20 0.31
PRKDC P78527 1/20 0.31
ATM Q13315 1/20 0.31
ATR Q13535 1/20 0.31
FLT1 P17948 1/20 0.31
FLT4 P35916 1/20 0.31
KDR P35968 1/20 0.31
NR1I2 O75469 1/20 0.30
SCN1B Q07699 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1631121 0.82 PSEN1 (0.38) S1PR3S1PR1SCN1ASCN5ASCN8A
SCHEMBL28772200 0.78 TRPV4 (0.33) S1PR3S1PR1S1PR4SCN1ASCN5A
SCHEMBL1632894 0.73 PSEN1 (0.42) PIK3CAMTORATR
SCHEMBL1631914 0.72 PSEN1 (0.39) S1PR3S1PR1S1PR4SCN1ASCN5A
SCHEMBL12762203 0.70 PSEN1 (0.38) S1PR3S1PR1SCN1ASCN5ASCN8A
SCHEMBL1632260 0.68 PSEN1 (0.53)
SCHEMBL1632245 0.67 PSEN1 (0.37) S1PR3S1PR1SCN1ASCN5ASCN8A
SCHEMBL1631232 0.67 SCN1A (0.41) S1PR3SCN1ASCN5ASCN8ATNF
SCHEMBL1632122 0.65 PSEN1 (0.43) SCN1ASCN5ASCN8APIK3CAMTOR
SCHEMBL1631897 0.65 PSEN1 (0.48) PIK3CAMTOR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-100378072-C Heterocyclic methyl sulfone derivative DAIICHI SEIYAKU CO (JP) 2008-04-02 CN disclosed