SCHEMBL28779254

SCHEMBL28779254

CC(C)(C)NC(=O)OC[C@H]1CCNC1

nearest known ligand 0.48

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CHRM3 P20309 13/20 0.48
SLC6A1 P30531 2/20 0.42
GABRA5 P31644 2/20 0.42
GABRB2 P47870 2/20 0.42
SLC6A12 P48065 2/20 0.42
SLC6A11 P48066 2/20 0.42
SLC6A13 Q9NSD5 2/20 0.42
GABRA1 P14867 1/20 0.42
GABRR1 P24046 1/20 0.42
GABRA4 P48169 1/20 0.42
CHRM2 P08172 5/20 0.39
CHRM1 P11229 5/20 0.39
HDAC1 Q13547 3/20 0.36
HDAC2 Q92769 3/20 0.36
HDAC3 O15379 2/20 0.36
CHRNB2 P17787 1/20 0.35
CHRNB4 P30926 1/20 0.35
CHRNA3 P32297 1/20 0.35
CHRNA4 P43681 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27917819 1.00 CHRM3 (0.48) CHRM3SLC6A1GABRA5GABRB2SLC6A12
SCHEMBL27789305 0.91 HDAC3 (0.44) CHRM3SLC6A1SLC6A11SLC6A13HDAC1
SCHEMBL27714539 0.91 HDAC3 (0.44) CHRM3SLC6A1SLC6A11SLC6A13HDAC1
SCHEMBL27810874 0.91 HDAC3 (0.44) CHRM3SLC6A1SLC6A11SLC6A13HDAC1
SCHEMBL1428636 0.90 CHRM3 (0.46) CHRM3CHRM2CHRM1HDAC1HDAC2
SCHEMBL1367746 0.87 HDAC1 (0.38) CHRM3CHRM2CHRM1HDAC1HDAC2
Hydrochloric Acid SCHEMBL22291356 0.85 HDAC1 (0.38) CHRM3CHRM2CHRM1HDAC1HDAC2
SCHEMBL25274161 0.85 CHRM3 (0.42) CHRM3CHRM2CHRM1HDAC1HDAC2
SCHEMBL27973838 0.81 EPHX1 (0.45)
SCHEMBL25518973 0.81 CNR2 (0.40) CHRM3CHRM2CHRM1HDAC1HDAC2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114761394-B Pyridine or pyrimidine derivative and preparation method and application thereof 浙江海正药业股份有限公司 2024-03-29 CN disclosed
CN-115916765-A Pyridine or pyrimidine derivative and preparation method and application thereof 浙江海正药业股份有限公司 2023-04-04 CN disclosed
CN-114761394-A Pyridine or pyrimidine derivative and preparation method and application thereof 浙江海正药业股份有限公司 2022-07-15 CN disclosed
CN-113924292-A Antimicrobial compounds and methods 库扎环球有限责任公司 2022-01-11 CN disclosed