SCHEMBL28779259

SCHEMBL28779259

Cc1nc(N2CCC(NC(=O)OC(C)(C)C)CC2)nc(C#N)c1Br

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CTSK P43235 2/20 0.46
JAK3 P52333 1/20 0.46
BTK Q06187 1/20 0.46
CKS1B P61024 1/20 0.43
SKP1 P63208 1/20 0.43
SKP2 Q13309 1/20 0.43
KCNA3 P22001 1/20 0.42
PDE10A Q9Y233 1/20 0.41
SUV39H2 Q9H5I1 7/20 0.39
RET P07949 1/20 0.39
PARP1 P09874 1/20 0.38
AAK1 Q2M2I8 1/20 0.38
OPRM1 P35372 1/20 0.38
OPRD1 P41143 1/20 0.38
OPRK1 P41145 1/20 0.38
OGFRL1 Q5TC84 1/20 0.38
DRD2 P14416 1/20 0.37
CNR1 P21554 1/20 0.37
CNR2 P34972 1/20 0.37
NSD2 O96028 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29770982 1.00 CTSK (0.46) CTSKJAK3BTKCKS1BSKP1
SCHEMBL23657173 0.84 BTK (0.42) CTSKJAK3BTKCKS1BSKP1
SCHEMBL24183332 0.84 JAK3 (0.41) CTSKJAK3BTKKCNA3PDE10A
SCHEMBL22389722 0.83 JAK3 (0.40) CTSKJAK3BTKCKS1BSKP1
SCHEMBL28779238 0.81 CKS1B (0.42) JAK3BTKCKS1BSKP1SKP2
SCHEMBL23657226 0.81 CKS1B (0.42) JAK3BTKCKS1BSKP1SKP2
SCHEMBL29771164 0.81 CKS1B (0.42) JAK3BTKCKS1BSKP1SKP2
SCHEMBL22389965 0.80 RET (0.40) JAK3BTKRET
SCHEMBL22389936 0.79 JAK3 (0.35) CTSKJAK3BTK
SCHEMBL22389941 0.79 JAK3 (0.35) CTSKJAK3BTKRET

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114761394-B Pyridine or pyrimidine derivative and preparation method and application thereof 浙江海正药业股份有限公司 2024-03-29 CN disclosed
CN-115916765-A Pyridine or pyrimidine derivative and preparation method and application thereof 浙江海正药业股份有限公司 2023-04-04 CN disclosed
CN-114761394-A Pyridine or pyrimidine derivative and preparation method and application thereof 浙江海正药业股份有限公司 2022-07-15 CN disclosed