SCHEMBL28782892

SCHEMBL28782892

COC(=O)N[C@@H](C(=O)N1CCC[C@H]1c1ncc(-c2cnc([C@@H]3CCCN3C(=O)O)[nH]2)[nH]1)c1ccccc1

nearest known ligand 0.61

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 11/20 0.61
CYP2C9 P11712 9/20 0.61
KCNH2 Q12809 3/20 0.61
NR1I2 O75469 2/20 0.61
ABCB11 O95342 1/20 0.61
OPRK1 P41145 1/20 0.61
CYP1A2 P05177 4/20 0.55
CYP2D6 P10635 3/20 0.54
CYP2C19 P33261 5/20 0.48
OPRM1 P35372 1/20 0.45
OPRD1 P41143 1/20 0.45
PRCP P42785 2/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15477464 0.95 CYP3A4 (0.69) CYP3A4CYP2C9KCNH2NR1I2ABCB11
SCHEMBL2959577 0.95 CYP3A4 (0.69) CYP3A4CYP2C9KCNH2NR1I2ABCB11
SCHEMBL27780306 0.94 CYP3A4 (0.60) CYP3A4CYP2C9KCNH2NR1I2ABCB11
SCHEMBL10177209 0.93 CYP3A4 (0.71) CYP3A4CYP2C9KCNH2NR1I2ABCB11
SCHEMBL19578082 0.93 CYP3A4 (0.68) CYP3A4CYP2C9KCNH2NR1I2ABCB11
SCHEMBL10177580 0.92 CYP3A4 (0.73) CYP3A4CYP2C9KCNH2NR1I2ABCB11
SCHEMBL17571146 0.92 CYP3A4 (0.73) CYP3A4CYP2C9KCNH2NR1I2ABCB11
SCHEMBL12174942 0.91 KCNH2 (0.63) CYP3A4CYP2C9KCNH2NR1I2ABCB11
SCHEMBL28814568 0.90 CYP3A4 (0.56) CYP3A4CYP2C9KCNH2NR1I2ABCB11
SCHEMBL12175043 0.90 CYP3A4 (0.63) CYP3A4CYP2C9KCNH2NR1I2ABCB11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101528232-B Hepatitis c virus inhibitors BRISTOL MYERS SQUIBB CO 2014-11-12 CN disclosed
CN-101528232-A Hepatitis C virus inhibitors BRISTOL MYERS SQUIBB CO (US) 2009-09-09 CN disclosed