SCHEMBL28814568

SCHEMBL28814568

COC(=O)N[C@@H](C(=O)N1CCC[C@H]1c1ncc(-c2cnc([C@@H]3CCCN3C(=O)OC(C)(C)C)[nH]2)[nH]1)c1ccccc1

nearest known ligand 0.56

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 9/20 0.56
CYP2C9 P11712 8/20 0.56
KCNH2 Q12809 3/20 0.56
NR1I2 O75469 2/20 0.56
ABCB11 O95342 1/20 0.56
OPRK1 P41145 1/20 0.56
CYP1A2 P05177 4/20 0.53
CYP2D6 P10635 3/20 0.53
HPGDS O60760 3/20 0.46
CYP2C19 P33261 5/20 0.45
PRCP P42785 3/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL691516 0.95 CYP3A4 (0.64) CYP3A4CYP2C9KCNH2NR1I2ABCB11
SCHEMBL27780306 0.93 CYP3A4 (0.60) CYP3A4CYP2C9KCNH2NR1I2ABCB11
SCHEMBL10254082 0.92 CYP3A4 (0.58) CYP3A4CYP2C9KCNH2NR1I2ABCB11
SCHEMBL27989781 0.92 KCNH2 (0.54) CYP3A4CYP2C9KCNH2NR1I2ABCB11
SCHEMBL690281 0.92 CYP3A4 (0.58) CYP3A4CYP2C9KCNH2NR1I2ABCB11
SCHEMBL690282 0.92 CYP3A4 (0.58) CYP3A4CYP2C9KCNH2NR1I2ABCB11
SCHEMBL27780307 0.91 KCNH2 (0.52) CYP3A4CYP2C9KCNH2NR1I2ABCB11
SCHEMBL28782892 0.90 CYP3A4 (0.61) CYP3A4CYP2C9KCNH2NR1I2ABCB11
SCHEMBL8750715 0.90 CYP3A4 (0.58) CYP3A4CYP2C9KCNH2NR1I2ABCB11
SCHEMBL6121525 0.90 CYP3A4 (0.58) CYP3A4CYP2C9KCNH2NR1I2ABCB11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101558059-B Hepatitis c virus inhibitors BRISTOL MYERS SQUIBB CO 2014-12-03 CN claimed
CN-101558059-B Hepatitis c virus inhibitors BRISTOL MYERS SQUIBB CO 2014-12-03 CN disclosed
CN-101998952-B Hepatitis c virus inhibitors BRISTOL-MYERS SQUIBB CO. (US) 2014-10-08 CN disclosed