SCHEMBL28784362

SCHEMBL28784362

CC(C)(C)C(=O)ON1CCCC(NC(=O)c2ccc(Cn3ncc4ccccc43)cc2)C1

nearest known ligand 0.42

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
AURKA O14965 3/20 0.41
AURKB Q96GD4 3/20 0.41
OPRM1 P35372 1/20 0.41
OPRK1 P41145 1/20 0.41
DRD2 P14416 2/20 0.41
DRD4 P21917 2/20 0.41
PKM P14618 1/20 0.41
MCHR1 Q99705 4/20 0.41
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40
NPC1 O15118 1/20 0.40
RAB9A P51151 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
CRHR1 P34998 1/20 0.40
CCR2 P41597 1/20 0.39
TSHR P16473 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3665804 0.85 USP30 (0.56)
SCHEMBL3638888 0.81 USP30 (0.54)
SCHEMBL4938421 0.81 USP30 (0.54)
SCHEMBL7756336 0.79 HDAC4 (0.51) DRD4PKMMEN1KMT2ANPC1
SCHEMBL27808340 0.78 PTAFR (0.47) MCHR1
SCHEMBL27808373 0.77 CRHR1 (0.40) AURKAAURKBDRD4MEN1KMT2A
SCHEMBL28787440 0.77 CRHR1 (0.40) AURKAAURKBDRD4MEN1KMT2A
Tert-Butyl Formate SCHEMBL28784363 0.75 HDAC4 (0.41) AURKAAURKBOPRK1NPC1RAB9A
SCHEMBL8366923 0.71 RECQL (0.60) MEN1KMT2ANPC1RAB9ASMN1; SMN2
SCHEMBL27759531 0.71 USP30 (0.49) MEN1KMT2AL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101778838-A Azacyclylbenzamide derivatives as histamine-3 antagonists WYETH CORP 2010-07-14 CN disclosed