SCHEMBL2878693

SCHEMBL2878693

Cc1c(N[C@H]2CCc3ccccc32)ccnc1Cl

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FADS1 O60427 1/20 0.48
PDPK1 O15530 1/20 0.48
CYP3A4 P08684 4/20 0.46
NSD2 O96028 2/20 0.46
KDM4E B2RXH2 1/20 0.46
MEN1 O00255 1/20 0.46
ALDH1A1 P00352 1/20 0.46
TP53 P04637 1/20 0.46
MAPT P10636 1/20 0.46
THRB P10828 1/20 0.46
TSHR P16473 1/20 0.46
MAPK1 P28482 1/20 0.46
CASP1 P29466 1/20 0.46
CDC25B P30305 1/20 0.46
RECQL P46063 1/20 0.46
BLM P54132 1/20 0.46
CASP7 P55210 1/20 0.46
KMT2A Q03164 1/20 0.46
SMN1; SMN2 Q16637 1/20 0.46
BRS3 P32247 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2350272 0.79 FADS1 (0.43) FADS1PDPK1CYP3A4NSD2KDM4E
SCHEMBL5691101 0.70 PDPK1 (0.53) FADS1PDPK1CYP3A4NSD2KDM4E
SCHEMBL783904 0.69 PFKFB3 (0.49) FADS1PDPK1CYP3A4NSD2KDM4E
SCHEMBL2476603 0.69 CYP3A4 (0.46) FADS1PDPK1CYP3A4NSD2KDM4E
SCHEMBL782435 0.69 FADS1 (0.55) FADS1PDPK1CYP3A4NSD2KDM4E
SCHEMBL20511289 0.69 FADS1 (0.55) FADS1PDPK1CYP3A4NSD2KDM4E
SCHEMBL26614814 0.69 FADS1 (0.51) FADS1PDPK1CYP3A4NSD2KDM4E
SCHEMBL26614621 0.69 FADS1 (0.51) FADS1PDPK1CYP3A4NSD2KDM4E
SCHEMBL26614619 0.69 FADS1 (0.51) FADS1PDPK1CYP3A4NSD2KDM4E
SCHEMBL782718 0.68 PFKFB3 (0.53) FADS1PDPK1MAOAMAOBPFKFB3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2049491-B1 HETEROARYL COMPOUNDS USEFUL AS INHIBITORS OF E1 ACTIVATING ENZYMES MILLENNIUM PHARM INC (US) 2010-10-20 EP disclosed