SCHEMBL2878752

SCHEMBL2878752

CC1CCC(C(=O)N(c2cc(-c3cccc(F)c3)sc2OC(=O)O)C2CCC(O)CC2)CC1

nearest known ligand 0.46

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
GRM5 P41594 1/20 0.35
S1PR1 P21453 1/20 0.34
FYN P06241 1/20 0.33
KDM4E B2RXH2 1/20 0.32
HTT P42858 1/20 0.32
ATM Q13315 1/20 0.32
JAK2 O60674 1/20 0.32
VCP P55072 1/20 0.32
OPRM1 P35372 1/20 0.31
POLB P06746 1/20 0.31
HSD17B1 P14061 2/20 0.31
HSD17B2 P37059 2/20 0.31
STK17B O94768 1/20 0.31
CDK2AP1 O14519 1/20 0.30
CHEK1 O14757 1/20 0.30
NR1I2 O75469 2/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2871309 0.93 GRM5 (0.33) GRM5S1PR1FYNKDM4EHTT
SCHEMBL2877206 0.92 KDM4E (0.38) KDM4EHTTATMOPRM1NR1I2
SCHEMBL2874240 0.92 KDM4E (0.38) KDM4EHTTATMOPRM1NR1I2
SCHEMBL2874208 0.92 KDM4E (0.38) KDM4EHTTATMOPRM1NR1I2
SCHEMBL2879111 0.92 IKBKB (0.37) KDM4EHTTATMPOLB
SCHEMBL2878751 0.88 NR1I2 (0.39) GRM5S1PR1FYNKDM4EHTT
SCHEMBL2876896 0.88 NR1I2 (0.31) NR1I2
SCHEMBL2879449 0.88 KDM4E (0.36) KDM4EHTTATMOPRM1
SCHEMBL2879323 0.86 KDM4E (0.38) KDM4EHTTATMVCPOPRM1
SCHEMBL2878858 0.86 KDM4E (0.39) KDM4EHTTATMVCP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1569929-B9 COMPOUNDS AND METHODS FOR THE TREATMENT OR PREVENTION OF FLAVIVIRUS INFECTIONS VIROCHEM PHARMA INC (CA) 2011-09-14 EP claimed
EP-1569929-B1 COMPOUNDS AND METHODS FOR THE TREATMENT OR PREVENTION OF FLAVIVIRUS INFECTIONS VIROCHEM PHARMA INC (CA) 2010-05-05 EP claimed