SCHEMBL28790280

SCHEMBL28790280

CC(=O)Oc1nc(C)sc1-c1ccccc1

nearest known ligand 0.73

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ALOX5 P09917 2/20 0.73
NTRK1 P04629 1/20 0.43
PTGS1 P23219 2/20 0.43
PTGS2 P35354 2/20 0.43
SMN1; SMN2 Q16637 2/20 0.41
ALDH1A1 P00352 2/20 0.41
KDM4E B2RXH2 1/20 0.41
HPGD P15428 1/20 0.41
HSD17B10 Q99714 1/20 0.41
GRM6 O15303 1/20 0.40
BACE1 P56817 1/20 0.40
FFAR4 Q5NUL3 1/20 0.39
MEN1 O00255 1/20 0.39
MAPT P10636 1/20 0.39
KMT2A Q03164 1/20 0.39
GAA P10253 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14631965 0.89 ALOX5 (0.57) ALOX5NTRK1PTGS1PTGS2SMN1; SMN2
SCHEMBL27824201 0.88 ALOX5 (0.56) ALOX5SMN1; SMN2KDM4EMEN1MAPT
SCHEMBL28786380 0.85 ALOX5 (0.54) ALOX5PTGS1PTGS2ALDH1A1GRM6
SCHEMBL27837187 0.85 ALOX5 (0.54) ALOX5PTGS1PTGS2SMN1; SMN2ALDH1A1
SCHEMBL9629544 0.84 ALOX5 (1.00) ALOX5SMN1; SMN2ALDH1A1KDM4EMEN1
SCHEMBL27803410 0.84 ALOX5 (0.73) ALOX5PTGS1PTGS2SMN1; SMN2ALDH1A1
SCHEMBL28790234 0.83 ALOX5 (0.52) ALOX5PTGS2SMN1; SMN2MAPTKMT2A
SCHEMBL27899608 0.83 ALOX5 (0.52) ALOX5PTGS2GAA
SCHEMBL27626587 0.83 ALOX5 (0.71) ALOX5SMN1; SMN2ALDH1A1KDM4EHPGD
SCHEMBL27817785 0.82 ALOX5 (0.55) ALOX5SMN1; SMN2ALDH1A1HPGDFFAR4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102164896-A Phenethylamide derivatives and their heterocyclic analogues ACTELION PHARMACEUTICALS LTD 2011-08-24 CN disclosed
CN-101965343-A 2-aza-bicyclo[2.2.1]heptane derivatives ACTELION PHARMACEUTICALS LTD 2011-02-02 CN disclosed