SCHEMBL28790508

SCHEMBL28790508

O=CC(CN1CCN(c2cccc(C(F)(F)F)c2)CC1)c1ccc(F)cc1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IGF1R P08069 1/20 0.58
ADRB2 P07550 1/20 0.52
ADRB1 P08588 1/20 0.52
ADRB3 P13945 1/20 0.52
ADRA1D P25100 1/20 0.52
ADRA1A P35348 1/20 0.52
ADRA1B P35368 1/20 0.52
SIGMAR1 Q99720 2/20 0.50
ALDH1A1 P00352 4/20 0.48
MAPT P10636 4/20 0.48
MEN1 O00255 3/20 0.48
KMT2A Q03164 3/20 0.48
MAPK1 P28482 2/20 0.48
GAA P10253 1/20 0.48
HTT P42858 1/20 0.48
KDM4E B2RXH2 4/20 0.48
LMNA P02545 3/20 0.48
CYP1A2 P05177 2/20 0.48
CYP3A4 P08684 2/20 0.48
CYP2D6 P10635 2/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27826229 0.90 IGF1R (0.57) IGF1RADRB2ADRB1ADRB3ADRA1D
SCHEMBL27845191 0.90 IGF1R (0.57) IGF1RADRB2ADRB1ADRB3ADRA1D
SCHEMBL27826235 0.90 IGF1R (0.54) IGF1RADRB2ADRB1ADRB3ADRA1D
SCHEMBL27940499 0.88 IGF1R (0.54) IGF1RADRB2ADRB1ADRB3ADRA1D
SCHEMBL27826192 0.86 IGF1R (0.53) IGF1RADRB2ADRB1ADRB3ADRA1D
SCHEMBL27845189 0.86 IGF1R (0.53) IGF1RADRB2ADRB1ADRB3ADRA1D
SCHEMBL27845382 0.84 IGF1R (0.53) IGF1RADRB2ADRB1ADRB3ADRA1D
SCHEMBL27845205 0.84 IGF1R (0.53) IGF1RADRB2ADRB1ADRB3ADRA1D
SCHEMBL28790506 0.83 IGF1R (0.60) IGF1RADRB2ADRB1ADRB3ADRA1D
SCHEMBL27826227 0.83 ALDH1A1 (0.53) IGF1RADRB2ADRB1ADRB3ADRA1D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101985438-A Substituted phenyl piperazinyl aralkylone derivatives and application thereof to preparation of analgesics JIANGSU NHWA PHARMACEUTICAL CO LTD 2011-03-16 CN claimed
CN-101985438-A Substituted phenyl piperazinyl aralkylone derivatives and application thereof to preparation of analgesics JIANGSU NHWA PHARMACEUTICAL CO LTD 2011-03-16 CN disclosed