SCHEMBL28790797

SCHEMBL28790797

Cc1ccc(C(=O)Cl)c(N)c1[N+](=O)[O-]

nearest known ligand 0.44

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 8/20 0.44
TDP1 Q9NUW8 3/20 0.44
TSHR P16473 6/20 0.40
CYP3A4 P08684 5/20 0.39
RECQL P46063 1/20 0.39
POLB P06746 2/20 0.37
HPGD P15428 1/20 0.37
ALOX15 P16050 1/20 0.36
MEN1 O00255 2/20 0.35
KMT2A Q03164 2/20 0.35
MAPT P10636 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1644833 0.85 ALDH1A1 (0.47) ALDH1A1TDP1TSHRCYP3A4RECQL
SCHEMBL11695700 0.83 ALDH1A1 (0.47) ALDH1A1TDP1TSHRCYP3A4POLB
SCHEMBL28061957 0.81 ALDH1A1 (0.46) ALDH1A1TDP1TSHRCYP3A4POLB
SCHEMBL27898207 0.80 ALDH1A1 (0.39) ALDH1A1TDP1TSHRCYP3A4HPGD
SCHEMBL27338694 0.79 ALDH1A1 (0.42) ALDH1A1TDP1TSHRPOLBHPGD
SCHEMBL8501106 0.79 ALDH1A1 (0.50) ALDH1A1TDP1TSHRCYP3A4RECQL
SCHEMBL28194935 0.78 MAPK14 (0.47) ALDH1A1TDP1TSHRMAPT
SCHEMBL11453634 0.78 MAPT (0.49) ALDH1A1TSHRCYP3A4RECQLPOLB
SCHEMBL28226522 0.78 ALDH1A1 (0.41) ALDH1A1TDP1TSHRPOLBHPGD
SCHEMBL14269307 0.78 ALDH1A1 (0.58) ALDH1A1TDP1TSHRCYP3A4RECQL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102050814-B Ester derivatives of dabigatran BEIJING MEIBEITA PHARMACEUTICAL RES INST CO LTD 2014-05-28 CN disclosed
CN-102050815-B Dabigatran ester derivatives as prodrug BEIJING MEIBEITA PHARMACEUTICAL RES CO LTD 2014-04-02 CN disclosed
CN-103420980-A Dabigatran derivatives BEIJING MEIBEITA DRUG RES CO LTD 2013-12-04 CN disclosed
CN-102050815-A Dabigatran ester derivatives as prodrug BEIJING MEIBEITA PHARMACEUTICAL RES INST CO LTD 2011-05-11 CN disclosed
CN-102050814-A Ester derivatives of dabigatran BEIJING MEIBEITA PHARMACEUTICAL RES INST CO LTD 2011-05-11 CN disclosed