SCHEMBL28794849

SCHEMBL28794849

COC(=O)c1ccc(OB(O)O)cc1Cl

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ABL1 P00519 1/20 0.45
JAK2 O60674 1/20 0.43
TYK2 P29597 1/20 0.43
CLPP Q16740 2/20 0.42
PDK2 Q15119 2/20 0.41
CA12 O43570 1/20 0.41
CA1 P00915 1/20 0.41
CA2 P00918 1/20 0.41
CA7 P43166 1/20 0.41
PDK4 Q16654 1/20 0.41
CA9 Q16790 1/20 0.41
CA14 Q9ULX7 1/20 0.41
MAPT P10636 3/20 0.41
RAB9A P51151 2/20 0.41
CYP1A2 P05177 2/20 0.41
CYP2C19 P33261 2/20 0.41
FLT1 P17948 2/20 0.41
FLT4 P35916 2/20 0.41
KDR P35968 2/20 0.41
KDM4E B2RXH2 3/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28081598 0.87 MEN1 (0.48) ABL1TYK2MAPTCYP1A2CYP2C19
SCHEMBL1180038 0.83 TYK2 (0.57) ABL1JAK2TYK2PDK2CA12
SCHEMBL30819021 0.82 CA12 (0.64) PDK2CA12CA1CA2CA7
SCHEMBL20987087 0.82 KDM4E (0.44) ABL1PDK2CA12CA1CA2
SCHEMBL28006591 0.82 CA12 (0.64) PDK2CA12CA1CA2CA7
SCHEMBL27853433 0.81 CPS1 (0.44) ABL1PDK2CA12CA1CA2
SCHEMBL21434767 0.81 PDK2 (0.47) ABL1JAK2TYK2PDK2CA12
SCHEMBL516293 0.79 ABL1 (0.46) ABL1JAK2TYK2PDK2CA12
SCHEMBL1014886 0.79 ALDH1A1 (0.53) ABL1JAK2TYK2PDK2CA12
SCHEMBL21447016 0.77 TDP1 (0.51) ABL1MAPTRAB9AKDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102711470-A Novel tricyclic compounds ABBOTT LAB 2012-10-03 CN disclosed
CN-102356068-A 2,3-diaryl- or heteroaryl-substituted 1,1,1-trifluoro-2-hydroxypropyl compounds HOFFMANN LA ROCHE 2012-02-15 CN disclosed