SCHEMBL28798205

SCHEMBL28798205

Fc1ccc(F)c2c1CCCN2

nearest known ligand 0.39

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.39
MEN1 O00255 1/20 0.39
ALDH1A1 P00352 1/20 0.39
TP53 P04637 1/20 0.39
GAA P10253 1/20 0.39
MAPT P10636 1/20 0.39
ALOX15 P16050 1/20 0.39
ALOX12 P18054 1/20 0.39
MPI P34949 1/20 0.39
HTT P42858 1/20 0.39
KMT2A Q03164 1/20 0.39
HSD17B10 Q99714 1/20 0.39
TDP1 Q9NUW8 1/20 0.39
PARP1 P09874 13/20 0.39
PRKD1 Q15139 1/20 0.35
NPC1 O15118 1/20 0.34
RAB9A P51151 1/20 0.34
SRC P12931 1/20 0.33
HTR2C P28335 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31159121 0.89 HTR2C (0.39) MEN1MAPTKMT2APARP1HTR2C
SCHEMBL11901340 0.84 PARP1 (0.44) KDM4EMEN1ALDH1A1TP53GAA
SCHEMBL11901695 0.79 PARP1 (0.43) KDM4EMEN1ALDH1A1TP53GAA
SCHEMBL5330428 0.79 PARP1 (0.49) KDM4EMAPTPARP1
SCHEMBL619582 0.75 PARP10 (0.37) HTR2C
SCHEMBL31159167 0.72 NOTUM (0.47) KDM4EMEN1ALDH1A1TP53GAA
SCHEMBL31393728 0.72 PARP10 (0.42) HTR2C
SCHEMBL14232642 0.71 ERN1 (0.35) HTR2C
SCHEMBL25374470 0.71 GRIA1 (0.45) KDM4EALDH1A1TP53GAAMAPT
SCHEMBL2260714 0.71 GRIA1 (0.41) KDM4EALDH1A1TP53GAAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102702044-A Carbocyclic and heterocyclic arylsulfones as gamma secretase inhibitors SCHERING CORP 2012-10-03 CN disclosed