SCHEMBL5330428

SCHEMBL5330428

O=C(O)c1ccc(F)c2c1NCCC2

nearest known ligand 0.49

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 16/20 0.49
KDM4E B2RXH2 1/20 0.36
MAPT P10636 1/20 0.36
RXRA P19793 2/20 0.36
RXRB P28702 2/20 0.36
RXRG P48443 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL621034 0.90 PARP1 (0.40) PARP1KDM4ERXRARXRBRXRG
SCHEMBL5328082 0.82 PARP1 (0.53) PARP1KDM4E
SCHEMBL5328612 0.81 PARP1 (0.39) PARP1KDM4EMAPT
SCHEMBL3950495 0.81 ALDH1A1 (0.49) PARP1KDM4EMAPT
SCHEMBL3943394 0.80 MEN1 (0.40) PARP1KDM4EMAPTRXRARXRB
SCHEMBL28798205 0.79 KDM4E (0.39) PARP1KDM4EMAPT
SCHEMBL5754704 0.75 CYP1A2 (0.44) PARP1MAPTRXRARXRBRXRG
SCHEMBL21465443 0.75 CYP1A2 (0.44) PARP1MAPTRXRARXRBRXRG
SCHEMBL6970151 0.75 PARP1 (0.39) PARP1KDM4EMAPTRXRARXRB
SCHEMBL11901340 0.73 PARP1 (0.44) PARP1KDM4EMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007028789-A1 QUINAZOLINE DERIVATIVES AS ANTIVIRAL AGENTS ISTITUTO DI RICERCHE DI BIOLOGIA MOLECOLARE P. ANGELETTI SPA (IT) 2007-03-15 WO disclosed