SCHEMBL28798385

SCHEMBL28798385

COc1cc2ncnc(Nc3ccnc(N4CCOCC4)c3)c2cc1N

nearest known ligand 0.56

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
EGFR P00533 7/20 0.56
KDR P35968 5/20 0.50
EPHA2 P29317 4/20 0.50
EPHB4 P54760 2/20 0.50
RET P07949 1/20 0.50
MAPK14 Q16539 4/20 0.49
SRC P12931 3/20 0.49
ERBB2 P04626 1/20 0.49
CLK1 P49759 1/20 0.48
ABCG2 Q9UNQ0 1/20 0.48
LCK P06239 1/20 0.47
PDE10A Q9Y233 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29713885 0.86 EGFR (0.49) EGFRKDREPHA2EPHB4MAPK14
SCHEMBL28798364 0.86 EGFR (0.49) EGFRKDREPHA2EPHB4MAPK14
SCHEMBL28798336 0.84 EGFR (0.59) EGFRKDREPHA2EPHB4MAPK14
SCHEMBL28798349 0.83 PDE10A (0.50) EGFRKDREPHA2EPHB4RET
SCHEMBL28950334 0.81 EGFR (0.47) EGFRKDREPHA2EPHB4MAPK14
SCHEMBL28798340 0.80 PDE10A (0.47) EGFRKDREPHA2EPHB4MAPK14
SCHEMBL28798405 0.80 PDE10A (0.47) EGFRKDREPHA2EPHB4MAPK14
SCHEMBL29713896 0.80 PDE10A (0.47) EGFRKDREPHA2EPHB4MAPK14
SCHEMBL161067 0.80 EGFR (0.63) EGFRKDRRETSRC
SCHEMBL29713893 0.79 EGFR (0.50) EGFRKDREPHA2EPHB4RET

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114835683-A Quinazoline-4, 6-diamine compound containing morpholinyl aromatic heterocycle and preparation method thereof 江苏食品药品职业技术学院 2022-08-02 CN disclosed