SCHEMBL2880023

SCHEMBL2880023

COc1ccnc(Cn2cccc(C(F)(F)F)c2=O)c1COc1ccc2nc(C)cc(-c3ncsc3Cl)c2c1

nearest known ligand 0.67

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
BDKRB2 P30411 6/20 0.67
CYP3A4 P08684 2/20 0.67
CYP2C19 P33261 1/20 0.67
PTGDR2 Q9Y5Y4 2/20 0.33
NR1H4 Q96RI1 1/20 0.31
SYK P43405 1/20 0.31
EIF4EBP1 Q13541 6/20 0.31
P2RX7 Q99572 2/20 0.31
RORC P51449 1/20 0.30
ATP1A1 P05023 1/20 0.30
ATP1B1 P05026 1/20 0.30
ATP1A3 P13637 1/20 0.30
ATP1B2 P14415 1/20 0.30
ATP4A P20648 1/20 0.30
ATP1A2 P50993 1/20 0.30
ATP4B P51164 1/20 0.30
ATP1B3 P54709 1/20 0.30
FXYD2 P54710 1/20 0.30
ATP1A4 Q13733 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2868604 0.93 BDKRB2 (0.76) BDKRB2CYP3A4CYP2C19EIF4EBP1RORC
SCHEMBL2875517 0.88 BDKRB2 (0.61) BDKRB2CYP3A4CYP2C19PTGDR2NR1H4
SCHEMBL2872135 0.88 BDKRB2 (0.52) BDKRB2CYP3A4CYP2C19SYKEIF4EBP1
SCHEMBL1564395 0.87 BDKRB2 (0.87) BDKRB2CYP3A4CYP2C19RORC
SCHEMBL2871993 0.81 BDKRB2 (0.48) BDKRB2CYP3A4CYP2C19PTGDR2NR1H4
SCHEMBL2868602 0.80 BDKRB2 (1.00) BDKRB2CYP3A4CYP2C19RORC
SCHEMBL13093047 0.80 BDKRB2 (0.90) BDKRB2CYP3A4CYP2C19RORC
SCHEMBL13146271 0.80 BDKRB2 (0.80) BDKRB2CYP3A4CYP2C19RORC
SCHEMBL12711960 0.80 BDKRB2 (0.88) BDKRB2CYP3A4CYP2C19RORC
SCHEMBL2874958 0.79 BDKRB2 (0.50) BDKRB2CYP3A4CYP2C19EIF4EBP1RORC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2144897-B1 8-OXY-QUINOLINE DERIVATIVES AS BRADYKININ B2 RECEPTOR MODULATORS JERINI AG (DE) 2010-10-20 EP claimed