SCHEMBL28801522

SCHEMBL28801522

COC(=O)c1ccc(OCCCN2CCOCC2)cc1O

nearest known ligand 0.62

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
LMNA P02545 2/20 0.62
MAOB P27338 10/20 0.62
MAPK1 P28482 2/20 0.55
HRH3 Q9Y5N1 2/20 0.55
ALDH1A1 P00352 1/20 0.55
CYP1A2 P05177 1/20 0.55
CHRM2 P08172 1/20 0.55
CHRM1 P11229 1/20 0.55
HTR2A P28223 1/20 0.55
SCN1A P35498 1/20 0.55
HTR2B P41595 1/20 0.55
KCNH2 Q12809 1/20 0.55
SCN2A Q99250 1/20 0.55
SIGMAR1 Q99720 1/20 0.55
SCN3A Q9NY46 1/20 0.55
USP2 O75604 1/20 0.54
KDR P35968 1/20 0.53
EPHX2 P34913 2/20 0.53
MET P08581 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27895327 0.87 MAOB (0.62) LMNAMAOBMAPK1HRH3ALDH1A1
SCHEMBL23425648 0.82 MAOB (0.70) LMNAMAOBALDH1A1
SCHEMBL28678935 0.81 MAOB (0.65) LMNAMAOBMAPK1HRH3ALDH1A1
SCHEMBL6042793 0.81 LMNA (0.53) LMNAHRH3ALDH1A1
SCHEMBL31385612 0.81 MEN1 (0.53) MAPK1HRH3ALDH1A1CYP1A2CHRM2
SCHEMBL21681940 0.81 KDM4E (0.55) LMNAMAPK1HRH3ALDH1A1CYP1A2
SCHEMBL27926267 0.80 MAOB (0.61) LMNAMAOBEPHX2
SCHEMBL30344157 0.80 NPC1 (0.59) LMNAALDH1A1
SCHEMBL27934406 0.80 EPHX2 (0.62) ALDH1A1EPHX2
SCHEMBL3454279 0.79 HRH3 (0.47) LMNAMAPK1HRH3ALDH1A1CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102746255-A Compound having anti-tumor activity, and preparation method and application thereof ANHUI UNIVERSITY OF TRADITIONAL CHINESE MEDCINE 2012-10-24 CN disclosed