SCHEMBL28801565

SCHEMBL28801565

COc1cc2ncc(C#N)c(O)c2cc1O

nearest known ligand 0.53

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
EGFR P00533 9/20 0.53
ERBB2 P04626 8/20 0.53
MAP2K1 Q02750 3/20 0.52
SRC P12931 10/20 0.51
GAK O14976 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15279141 0.91 EGFR (0.62) EGFRERBB2MAP2K1SRCGAK
SCHEMBL4743551 0.87 SRC (0.51) EGFRERBB2MAP2K1SRCGAK
SCHEMBL28945823 0.86 EGFR (0.51) EGFRERBB2MAP2K1SRCGAK
SCHEMBL4950543 0.86 SRC (0.55) EGFRERBB2MAP2K1SRC
SCHEMBL20775350 0.86 EGFR (0.51) EGFRERBB2MAP2K1SRCGAK
SCHEMBL4294162 0.83 EGFR (0.51) EGFRERBB2MAP2K1SRCGAK
SCHEMBL13427130 0.81 EGFR (0.53) EGFRERBB2MAP2K1SRCGAK
SCHEMBL4786042 0.81 SRC (0.63) EGFRERBB2MAP2K1SRCGAK
SCHEMBL4741688 0.81 MAP2K1 (0.54) EGFRERBB2MAP2K1SRC
SCHEMBL22589792 0.80 SRC (0.56) EGFRERBB2MAP2K1SRCGAK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103012367-A Quinoline derivative UNIV PEKING FOUNDER GROUP CO 2013-04-03 CN disclosed
CN-103012368-A Quinoline derivative UNIV PEKING FOUNDER GROUP CO 2013-04-03 CN disclosed