SCHEMBL2880434

SCHEMBL2880434

CC(C)(C)[Si](C)(C)OC[C@H]1CC[C@@](Nc2ncnc3[nH]c(-c4cccc(Cl)c4)nc23)(O[Si](C)(C)C(C)(C)C)C1

nearest known ligand 0.37

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 1/20 0.37
MGAM O43451 1/20 0.34
GAA P10253 1/20 0.34
SI P14410 1/20 0.34
MGAM2 Q2M2H8 1/20 0.34
STK4 Q13043 1/20 0.34
STK3 Q13188 1/20 0.34
ADORA3 P0DMS8 1/20 0.33
ADORA2A P29274 1/20 0.33
ADORA2B P29275 1/20 0.33
ADORA1 P30542 1/20 0.33
KIT P10721 1/20 0.32
PARP1 P09874 1/20 0.32
MET P08581 1/20 0.31
KDR P35968 1/20 0.31
MAP4K4 O95819 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL783045 0.75 ADORA3 (0.38) GSK3BMGAMGAASIMGAM2
SCHEMBL796841 0.69 GSK3B (0.39) GSK3BMGAMGAASIMGAM2
SCHEMBL796842 0.69 GSK3B (0.39) GSK3BMGAMGAASIMGAM2
SCHEMBL805371 0.64 NAE1 (0.45) GSK3BSTK4STK3ADORA3ADORA2A
SCHEMBL783584 0.63 PARP1 (0.53) GSK3BMGAMGAASIMGAM2
SCHEMBL15007274 0.62 GSK3B (0.46) GSK3BMGAMGAASIMGAM2
Hydrochloric Acid SCHEMBL8595784 0.61 MAP4K4 (0.54) GSK3BMGAMGAASIMGAM2
SCHEMBL783619 0.60 NAE1 (0.61)
SCHEMBL15007272 0.60 GSK3B (0.46) GSK3BMGAMGAASIMGAM2
SCHEMBL3332631 0.54 MGAM (0.74) MGAMGAASIMGAM2ADORA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2049491-B1 HETEROARYL COMPOUNDS USEFUL AS INHIBITORS OF E1 ACTIVATING ENZYMES MILLENNIUM PHARM INC (US) 2010-10-20 EP disclosed