SCHEMBL28806102

SCHEMBL28806102

O=C(O)c1ccc(CNC(=O)c2cc(-c3ccccc3)nc3ccccc23)cc1

nearest known ligand 0.83

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TACR3 P29371 2/20 0.83
KDM4E B2RXH2 5/20 0.72
MEN1 O00255 1/20 0.72
POLB P06746 1/20 0.72
KMT2A Q03164 1/20 0.72
HDAC1 Q13547 2/20 0.67
ALDH1A1 P00352 5/20 0.66
TSHR P16473 1/20 0.65
LMNA P02545 5/20 0.65
SMN1; SMN2 Q16637 2/20 0.65
MAPK1 P28482 1/20 0.65
HTT P42858 2/20 0.64
NPC1 O15118 1/20 0.64
TP53 P04637 1/20 0.64
RAB9A P51151 1/20 0.64
TDP1 Q9NUW8 1/20 0.61
HPGD P15428 1/20 0.61
PDE10A Q9Y233 1/20 0.60
PTGER4 P35408 1/20 0.60
CYP3A4 P08684 1/20 0.60

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6450086 0.91 TACR3 (1.00) TACR3KDM4EMEN1POLBKMT2A
SCHEMBL28806105 0.89 TACR3 (0.76) TACR3KDM4EMEN1POLBKMT2A
SCHEMBL29271531 0.86 TACR3 (0.71) TACR3KDM4EMEN1POLBKMT2A
SCHEMBL6447321 0.82 TACR3 (0.81) TACR3KDM4EMEN1POLBKMT2A
SCHEMBL28511608 0.81 MAPT (0.82) TACR3KDM4EMEN1POLBKMT2A
SCHEMBL6630664 0.81 TACR3 (0.72) TACR3KDM4EMEN1POLBKMT2A
SCHEMBL10391576 0.81 TACR3 (0.76) TACR3KDM4EMEN1POLBKMT2A
SCHEMBL6447770 0.81 TACR3 (0.75) TACR3KDM4EMEN1POLBKMT2A
SCHEMBL8689228 0.80 DHODH (0.82) KDM4EPOLBKMT2AALDH1A1LMNA
SCHEMBL28806099 0.80 TACR3 (0.62) TACR3KDM4EMEN1POLBKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114890947-B Aromatic heterocyclic compound containing quinoline structural unit, and preparation method and application thereof 郑州大学 2024-07-16 CN disclosed
CN-114890947-A Aromatic heterocyclic compound containing quinoline structural unit and preparation method and application thereof 郑州大学 2022-08-12 CN disclosed