SCHEMBL28807635

SCHEMBL28807635

Cc1cc(C)cc(CC(c2cccc(Cl)c2)c2nc(-c3ccc(CNCCC(=O)O)cc3)no2)c1

nearest known ligand 0.48

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
PTPN1 P18031 6/20 0.48
S1PR1 P21453 4/20 0.45
FFAR1 O14842 2/20 0.42
S1PR3 Q99500 3/20 0.40
KMT2A Q03164 1/20 0.39
S1PR4 O95977 1/20 0.39
S1PR5 Q9H228 1/20 0.39
TP53 P04637 1/20 0.38
HDAC1 Q13547 1/20 0.37
HDAC8 Q9BY41 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9103709 0.92 S1PR1 (0.55) PTPN1S1PR1FFAR1S1PR3S1PR4
SCHEMBL27938780 0.90 PTPN1 (0.48) PTPN1S1PR1FFAR1HDAC1HDAC8
SCHEMBL27938890 0.90 PTPN1 (0.49) PTPN1S1PR1FFAR1S1PR3TP53
SCHEMBL27920250 0.89 PTPN1 (0.44) PTPN1S1PR1S1PR3KMT2AS1PR4
SCHEMBL27938775 0.88 PTPN1 (0.44) PTPN1S1PR1FFAR1S1PR3KMT2A
SCHEMBL27920264 0.88 PTPN1 (0.46) PTPN1S1PR1FFAR1HDAC1HDAC8
SCHEMBL27938944 0.87 TP53 (0.47) PTPN1S1PR1FFAR1S1PR3KMT2A
SCHEMBL28805778 0.85 PTPN1 (0.47) PTPN1S1PR1FFAR1TP53HDAC1
SCHEMBL9100995 0.84 PTPN1 (0.47) PTPN1S1PR1FFAR1TP53HDAC1
SCHEMBL9101572 0.83 FFAR1 (0.50) PTPN1S1PR1FFAR1S1PR3TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103338766-A Oxadiazole derivatives as sphingosine 1-phosphate (S1P) receptor modulators ALLERGAN INC 2013-10-02 CN claimed